SCHEMBL514275

SCHEMBL514275

CS(=O)(=O)c1ccc(I)cc1

nearest known ligand 0.56

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ENPP2 Q13822 2/20 0.56
CA1 P00915 2/20 0.50
CA2 P00918 2/20 0.50
MMP1 P03956 1/20 0.50
MMP2 P08253 1/20 0.50
MMP9 P14780 1/20 0.50
MMP8 P22894 1/20 0.50
MMP13 P45452 1/20 0.50
F2 P00734 2/20 0.47
PRSS1 P07477 2/20 0.47
PRSS2 P07478 2/20 0.47
PRSS3 P35030 2/20 0.47
RAPGEF4 Q8WZA2 1/20 0.47
PTGS2 P35354 5/20 0.46
CCR2 P41597 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2376239 0.85 ENPP2 (0.72) ENPP2PTGS2
SCHEMBL8658099 0.80 PTGS2 (0.72) PTGS2
SCHEMBL8974192 0.80 PTGS2 (0.44) ENPP2PTGS2
SCHEMBL17642663 0.79 CA1 (0.46) ENPP2CA1CA2MMP1MMP2
SCHEMBL7677302 0.77 PTGS2 (0.62) ENPP2CA2PTGS2
SCHEMBL896933 0.77 RAPGEF4 (0.56) CA1CA2MMP1MMP2MMP9
SCHEMBL17548700 0.77 ENPP2 (0.62) ENPP2PTGS2
SCHEMBL13662414 0.77 CA1 (0.42) CA1CA2MMP1MMP2MMP9
SCHEMBL10300269 0.77 PTGS2 (0.62) ENPP2CA2PTGS2
SCHEMBL24899771 0.75 F2 (0.44) ENPP2CA1CA2MMP1MMP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 93 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117088909-A Method for producing aryltrimethylstannane compound 上海致同建设工程科技有限公司 2023-11-21 CN claimed
US-12325696-B2 Indazole derivative, preparation method therefor, and pharmaceutical application thereof JIANGSU HENGRUI MEDICINE CO., LTD. (CN) 2025-06-10 US disclosed
CN-119320379-A Indazole derivative, preparation method and medical application thereof 江苏恒瑞医药股份有限公司 2025-01-17 CN disclosed
CN-113874367-B Indazole derivative, preparation method and medical application thereof 江苏恒瑞医药股份有限公司 2024-09-13 CN disclosed
US-20240239746-A1 PREPARATION METHOD FOR PYRROLE AMIDE COMPOUND SUNSHINE LAKE PHARMA CO., LTD. (CN) 2024-07-18 US disclosed
CN-115246785-B Process for preparing pyrrole amide compounds 年衍药业(珠海)有限公司 2024-03-26 CN disclosed
EP-4332091-A1 PREPARATION METHOD FOR PYRROLE AMIDE COMPOUND Sunshine Lake Pharma Co., Ltd. (CN) 2024-03-06 EP disclosed
CN-117088909-A Method for producing aryltrimethylstannane compound 上海致同建设工程科技有限公司 2023-11-21 CN disclosed
CN-111170991-B Antiproliferative compounds and methods of synthesis thereof 细胞基因公司 2023-10-31 CN disclosed
EP-3594211-B1 ANTIPROLIFERATIVE COMPOUNDS AND METHODS OF USE THEREOF CELGENE CORP (US) 2023-10-25 EP disclosed
CN-101415716-A Condensed imidazole derivatives as aldosterone synthase inhibitors SPEEDEL EXPERIMENTA AG (CH) 2009-04-22 CN disclosed
EP-1385508-B1 DIPEPTIDYL PEPTIDASE INHIBITORS FOR THE TREATMENT OR PREVENTION OF DIABETES MERCK & CO INC (US) 2008-05-21 EP disclosed
WO-2008041053-A2 INHIBITORS OF VEGF RECEPTOR AND HGF RECEPTOR SIGNALING METHYLGENE, INC. (CA) 2008-04-10 WO disclosed
WO-2008035209-A2 INHIBITORS OF PROTEIN TYROSINE KINASE ACTIVITY METHYLGENE INC. (CA) 2008-03-27 WO disclosed
CN-1028521-C Therapeutic agents BOOTS CO PLC (GB) 1995-05-24 CN disclosed
EP-0536151-B1 ORTHOSUBSTITUTED BIPHENYL GUANIDINE DERIVATIVES AND ANTIDIABETIC OR HYPOGLYCAEMIC AGENTS CONTAINING THEM BOOTS CO PLC (GB) 1994-09-14 EP disclosed
US-5302720-A Biphenyl-substituted guanidine derivatives useful as hypoglycaemic agents THE BOOTS COMPANY (GB) 1994-04-12 US disclosed
CN-1072173-A Therapeutical agent BOOTS CO PLC (GB) 1993-05-19 CN disclosed
EP-0536151-A1 ORTHOSUBSTITUTED BIPHENYL GUANIDINE DERIVATIVES AND ANTIDIABETIC OR HYPOGLYCAEMIC AGENTS CONTAINING THEM. BOOTS CO PLC (GB) 1993-04-14 EP disclosed
WO-1992000273-A1 ORTHOSUBSTITUTED BIPHENYL AMIDINE AND BIPHENYL GUANIDINE DERIVATIVES AND ANTIDIABETIC OR HYPOGLYCAEMIC AGENTS CONTAINING THEM THE BOOTS COMPANY PLC (GB) 1992-01-09 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12325696-B2 Indazole derivative, preparation method therefor, and pharmaceutical application thereof CYP19A1, HSD17B11, CYP51A1 ENPP2 3969/4885CA1 4362/4885CA2 4308/4885
US-20240239746-A1 PREPARATION METHOD FOR PYRROLE AMIDE COMPOUND HPGDS, HRH4, FAAH ENPP2 3404/4885CA1 3225/4885CA2 3693/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.