SCHEMBL8974249

SCHEMBL8974249

CS(=O)(=O)c1ccc(C2=CCC=C2c2ccc(Cl)c(C(F)(F)F)c2)cc1

nearest known ligand 0.57

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 14/20 0.57
NOTUM Q6P988 1/20 0.49
KIF11 P52732 1/20 0.48
TSHR P16473 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
CCR2 P41597 1/20 0.44
PTGS1 P23219 4/20 0.42
SCN9A Q15858 1/20 0.40
POLB P06746 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8974589 0.90 KIF11 (0.51) PTGS2KIF11PTGS1SCN9A
SCHEMBL8974191 0.88 KIF11 (0.55) PTGS2KIF11PTGS1
SCHEMBL8974570 0.87 PTGS2 (0.57) PTGS2NOTUMKIF11TSHRSMN1; SMN2
SCHEMBL8973789 0.85 KIF11 (0.49) PTGS2NOTUMKIF11PTGS1
SCHEMBL8974287 0.85 KIF11 (0.56) PTGS2KIF11PTGS1
SCHEMBL9118144 0.84 PTGS2 (0.62) PTGS2NOTUMKIF11TSHRSMN1; SMN2
SCHEMBL8974226 0.83 PTGS2 (0.60) PTGS2PTGS1
SCHEMBL8973748 0.83 KIF11 (0.72) PTGS2KIF11PTGS1
SCHEMBL8973743 0.83 KIF11 (0.52) PTGS2KIF11PTGS1
SCHEMBL8974142 0.82 PTGS2 (0.59) PTGS2KIF11PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5576339-A Pyridyl substituted cyclopentadienes for the treatment of inflamation HUANG HORNG-CHIH (US) 1996-11-19 US disclosed
WO-1995030656-A1 SUBSTITUTED CYCLOPENTADIENYL COMPOUNDS FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1995-11-16 WO disclosed
US-5418254-A Side effect reduction G. D. SEARLE & CO. (US) 1995-05-23 US disclosed