SCHEMBL8974287

SCHEMBL8974287

CS(=O)(=O)c1ccc(C2=CCC=C2c2ccc(F)c(C(F)(F)F)c2)cc1

nearest known ligand 0.56

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 2/20 0.56
PTGS2 P35354 17/20 0.51
PTGS1 P23219 4/20 0.42
ELANE P08246 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8973748 0.89 KIF11 (0.72) KIF11PTGS2PTGS1
SCHEMBL8974191 0.89 KIF11 (0.55) KIF11PTGS2PTGS1
SCHEMBL8973789 0.86 KIF11 (0.49) KIF11PTGS2PTGS1
SCHEMBL8974152 0.86 KIF11 (0.56) KIF11PTGS2PTGS1
SCHEMBL8974249 0.85 PTGS2 (0.57) KIF11PTGS2PTGS1
SCHEMBL8974382 0.84 PTGS2 (0.60) KIF11PTGS2PTGS1
SCHEMBL8973743 0.84 KIF11 (0.52) KIF11PTGS2PTGS1
SCHEMBL9118944 0.83 PTGS2 (0.65) KIF11PTGS2PTGS1ELANE
SCHEMBL8974106 0.83 PTGS2 (0.48) KIF11PTGS2PTGS1
SCHEMBL8974589 0.83 KIF11 (0.51) KIF11PTGS2PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5576339-A Pyridyl substituted cyclopentadienes for the treatment of inflamation HUANG HORNG-CHIH (US) 1996-11-19 US disclosed
WO-1995030656-A1 SUBSTITUTED CYCLOPENTADIENYL COMPOUNDS FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1995-11-16 WO disclosed
US-5418254-A Side effect reduction G. D. SEARLE & CO. (US) 1995-05-23 US disclosed