SCHEMBL8973789

SCHEMBL8973789

Cc1ccc(C2=CCC=C2c2ccc(S(C)(=O)=O)cc2)cc1C(F)(F)F

nearest known ligand 0.49

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 2/20 0.49
PTGS2 P35354 15/20 0.45
PTGS1 P23219 3/20 0.42
NR1H2 P55055 1/20 0.41
PDE3B Q13370 1/20 0.39
PDE3A Q14432 1/20 0.39
NOTUM Q6P988 1/20 0.39
CYP2C9 P11712 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8973743 0.89 KIF11 (0.52) KIF11PTGS2PTGS1NR1H2CYP2C9
SCHEMBL8974191 0.89 KIF11 (0.55) KIF11PTGS2PTGS1NR1H2
SCHEMBL8974532 0.88 KIF11 (0.48) KIF11PTGS2PTGS1PDE3BPDE3A
SCHEMBL8974287 0.86 KIF11 (0.56) KIF11PTGS2PTGS1
SCHEMBL8974249 0.85 PTGS2 (0.57) KIF11PTGS2PTGS1NOTUM
SCHEMBL27561072 0.84 KIF11 (0.67) KIF11PTGS2PTGS1NR1H2NOTUM
SCHEMBL8973748 0.84 KIF11 (0.72) KIF11PTGS2PTGS1
SCHEMBL6749827 0.83 KIF11 (0.43) KIF11PTGS2PTGS1NR1H2PDE3B
SCHEMBL9119695 0.83 PTGS2 (0.61) KIF11PTGS2PTGS1NR1H2PDE3B
SCHEMBL8974106 0.83 PTGS2 (0.48) KIF11PTGS2PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5576339-A Pyridyl substituted cyclopentadienes for the treatment of inflamation HUANG HORNG-CHIH (US) 1996-11-19 US disclosed
WO-1995030656-A1 SUBSTITUTED CYCLOPENTADIENYL COMPOUNDS FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1995-11-16 WO disclosed
US-5418254-A Side effect reduction G. D. SEARLE & CO. (US) 1995-05-23 US disclosed