SCHEMBL8974258

SCHEMBL8974258

COC(=O)C1(C(=O)OC)C=C(c2ccc(F)cc2)C(c2ccc(S(C)(=O)=O)nc2)=C1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 4/20 0.41
PTGS1 P23219 3/20 0.41
POLQ O75417 1/20 0.37
GPR55 Q9Y2T6 3/20 0.36
CTSK P43235 1/20 0.36
CA12 O43570 1/20 0.36
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
CA9 Q16790 1/20 0.36
LMNA P02545 1/20 0.35
POLB P06746 1/20 0.35
CCR1 P32246 2/20 0.35
CDK9 P50750 1/20 0.35
MAPK1 P28482 1/20 0.35
GPR119 Q8TDV5 1/20 0.34
PIK3CD O00329 1/20 0.34
PIP5K1C O60331 1/20 0.34
PIK3CB P42338 1/20 0.34
PI4KA P42356 1/20 0.34
PIK3CG P48736 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8974231 0.90 CA9 (0.46) PTGS2PTGS1GPR55CA12CA1
SCHEMBL8974628 0.88 PTGS2 (0.43) PTGS2PTGS1GPR55CTSKLMNA
SCHEMBL8973759 0.87 POLB (0.41) PTGS2POLQCTSKPOLBGPR119
SCHEMBL8974198 0.82 PTGS2 (0.61) PTGS2PTGS1
SCHEMBL8974381 0.82 PTGS2 (0.47) PTGS2PTGS1GPR55CDK9PIK3CD
SCHEMBL8974452 0.81 PTGS2 (0.44) PTGS2PTGS1GPR119PI4KBKDM4E
SCHEMBL8974101 0.80 PTGS2 (0.47) PTGS2PTGS1
SCHEMBL8974505 0.80 PTGS2 (0.43) PTGS2PTGS1CDK9KDM4ENPC1
SCHEMBL9117440 0.80 PTGS2 (0.66) PTGS2PTGS1GPR55CTSKCDK9
SCHEMBL8974426 0.80 POLQ (0.36) PTGS2PTGS1POLQCTSKCA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5576339-A Pyridyl substituted cyclopentadienes for the treatment of inflamation HUANG HORNG-CHIH (US) 1996-11-19 US disclosed
WO-1995030656-A1 SUBSTITUTED CYCLOPENTADIENYL COMPOUNDS FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1995-11-16 WO disclosed
US-5418254-A Side effect reduction G. D. SEARLE & CO. (US) 1995-05-23 US disclosed