SCHEMBL8974452

SCHEMBL8974452

COC(=O)C1(C(=O)OC)C=C(c2ccc(S(C)(=O)=O)cc2)C(c2ccc(F)nc2)=C1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 6/20 0.44
PTGS1 P23219 4/20 0.44
MMP2 P08253 1/20 0.41
MMP9 P14780 1/20 0.41
MMP13 P45452 1/20 0.41
KCNH2 Q12809 2/20 0.38
FBP1 P09467 1/20 0.37
KDM4E B2RXH2 1/20 0.37
NPC1 O15118 1/20 0.37
ALDH1A1 P00352 1/20 0.37
GLA P06280 1/20 0.37
RAB9A P51151 1/20 0.37
LRRK2 Q5S007 2/20 0.36
GPR119 Q8TDV5 1/20 0.36
MAP4K4 O95819 2/20 0.36
PIK3CA P42336 1/20 0.36
MINK1 Q8N4C8 1/20 0.36
PI4KB Q9UBF8 1/20 0.36
CSF1R P07333 2/20 0.36
LGMN Q99538 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8974835 0.90 CA1 (0.44) PTGS2PTGS1MMP2MMP9MMP13
SCHEMBL9117985 0.87 KCNH2 (0.51) PTGS2PTGS1KCNH2MAP4K4PIK3CA
SCHEMBL8974198 0.84 PTGS2 (0.61) PTGS2PTGS1
SCHEMBL8974783 0.82 PTGS2 (0.47) PTGS2PTGS1GPR119
SCHEMBL8974180 0.82 PTGS2 (0.50) PTGS2PTGS1MMP2MMP9MMP13
SCHEMBL8974088 0.82 PTGS2 (0.50) PTGS2PTGS1MMP2MMP9MMP13
SCHEMBL8974837 0.81 PTGS2 (0.43) PTGS2PTGS1ALDH1A1
SCHEMBL8974258 0.81 PTGS2 (0.41) PTGS2PTGS1KDM4ENPC1ALDH1A1
SCHEMBL8974101 0.80 PTGS2 (0.47) PTGS2PTGS1
SCHEMBL8974812 0.80 PTGS2 (0.49) PTGS2PTGS1MMP2MMP9MMP13

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5576339-A Pyridyl substituted cyclopentadienes for the treatment of inflamation HUANG HORNG-CHIH (US) 1996-11-19 US disclosed
WO-1995030656-A1 SUBSTITUTED CYCLOPENTADIENYL COMPOUNDS FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1995-11-16 WO disclosed
US-5418254-A Side effect reduction G. D. SEARLE & CO. (US) 1995-05-23 US disclosed