SCHEMBL8974294

SCHEMBL8974294

CCC1(CC)C=C(c2ccncc2)C(c2ccc(S(N)(=O)=O)cc2)=C1

nearest known ligand 0.50

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CA2 P00918 13/20 0.50
CA1 P00915 7/20 0.50
CA9 Q16790 8/20 0.46
CA12 O43570 7/20 0.46
LRRK2 Q5S007 3/20 0.45
IKBKB O14920 1/20 0.43
CHUK O15111 1/20 0.43
IKBKE Q14164 1/20 0.43
CA7 P43166 2/20 0.42
CA5A P35218 1/20 0.42
CA5B Q9Y2D0 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.41
NAMPT P43490 1/20 0.40
ALOX5 P09917 1/20 0.40
TSHR P16473 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8974089 0.87 PTGS2 (0.46) SMN1; SMN2ALOX5
SCHEMBL8974325 0.85 CA2 (0.50) CA2CA1CA9CA12LRRK2
SCHEMBL8974901 0.85 CA2 (0.50) CA2CA1CA9CA12LRRK2
SCHEMBL8974279 0.84 PTGS2 (0.55) CA2CA9CA12
SCHEMBL8973810 0.84 PTGS2 (0.55) CA2CA1CA9CA12CA7
SCHEMBL8974811 0.83 CA2 (0.54) CA2CA1CA9CA12LRRK2
SCHEMBL8974424 0.83 KIF11 (0.62) CA2CA1CA9CA12CA7
SCHEMBL8974520 0.80 CA2 (0.54) CA2CA1CA9CA12IKBKB
SCHEMBL8974376 0.80 PTGS2 (0.45) CA2CA1CA9CA12CA7
SCHEMBL8974140 0.79 KCNH2 (0.44) CA2CA1CA9CA12CA7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5576339-A Pyridyl substituted cyclopentadienes for the treatment of inflamation HUANG HORNG-CHIH (US) 1996-11-19 US disclosed
WO-1995030656-A1 SUBSTITUTED CYCLOPENTADIENYL COMPOUNDS FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1995-11-16 WO disclosed
US-5418254-A Side effect reduction G. D. SEARLE & CO. (US) 1995-05-23 US disclosed