SCHEMBL9117985

SCHEMBL9117985

COC(=O)C1(C(=O)OC)C=C(c2ccc(S(C)(=O)=O)cc2)C(c2ccc(C(F)(F)F)nc2)=C1

nearest known ligand 0.51

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 2/20 0.51
MAP4K4 O95819 1/20 0.51
PIK3CA P42336 1/20 0.51
MINK1 Q8N4C8 1/20 0.51
PI4KB Q9UBF8 1/20 0.51
PTGS2 P35354 14/20 0.43
PTGS1 P23219 6/20 0.43
TRPV3 Q8NET8 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8973691 0.91 CA1 (0.43) KCNH2MAP4K4PIK3CAMINK1PI4KB
SCHEMBL8974452 0.87 PTGS2 (0.44) KCNH2MAP4K4PIK3CAMINK1PI4KB
SCHEMBL8975759 0.85 PTGS2 (0.50) PTGS2PTGS1
SCHEMBL8974421 0.83 PTGS2 (0.43) KCNH2PTGS2PTGS1
SCHEMBL8974697 0.82 KCNH2 (0.54) KCNH2MAP4K4PIK3CAMINK1PI4KB
SCHEMBL8974336 0.82 KCNH2 (0.54) KCNH2MAP4K4PIK3CAMINK1PI4KB
SCHEMBL8973759 0.81 POLB (0.41) KCNH2MAP4K4PIK3CAMINK1PI4KB
SCHEMBL8974291 0.81 KCNH2 (0.53) KCNH2MAP4K4PIK3CAMINK1PI4KB
SCHEMBL8974117 0.81 PTGS2 (0.40) PTGS2PTGS1
SCHEMBL8974198 0.81 PTGS2 (0.61) PTGS2PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1995030656-A1 SUBSTITUTED CYCLOPENTADIENYL COMPOUNDS FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1995-11-16 WO disclosed
US-5418254-A Side effect reduction G. D. SEARLE & CO. (US) 1995-05-23 US disclosed