SCHEMBL8975300

SCHEMBL8975300

CCCC(NNC(=O)OC(C)(C)C)C(O)C(F)(F)F

nearest known ligand 0.40

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
APLNR P35414 1/20 0.40
CTSK P43235 14/20 0.38
CTSS P25774 2/20 0.38
CA1 P00915 2/20 0.36
CA7 P43166 2/20 0.36
CA2 P00918 1/20 0.36
MEN1 O00255 1/20 0.35
GAA P10253 1/20 0.35
KMT2A Q03164 1/20 0.35
CA12 O43570 1/20 0.34
CA14 Q9ULX7 1/20 0.34
CYP2D6 P10635 1/20 0.33
CTSL P07711 1/20 0.32
CTSB P07858 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Benzene SCHEMBL5809252 0.81 CTSK (0.46) CTSKCTSSCA1CA7CA2
SCHEMBL2681437 0.74 CTSK (0.43) APLNRCTSKCTSSCA1CA7
SCHEMBL8543748 0.74 CTSK (0.43) APLNRCTSKCTSSCA1CA7
SCHEMBL2681435 0.74 CTSK (0.43) APLNRCTSKCTSSCA1CA7
SCHEMBL8041100 0.73 CA1 (0.55) CTSKCTSSCA1CA7CA2
SCHEMBL15247712 0.72 CTSK (0.49) CTSKCTSSCA1CA7CA2
SCHEMBL12011309 0.72 CA1 (0.44) APLNRCTSKCTSSCA1CA7
SCHEMBL5154942 0.71 CA1 (0.53) CTSKCTSSCA1CA7CA2
SCHEMBL20583908 0.71 APLNR (0.46) APLNRCTSKCTSSCA1CA7
SCHEMBL27859377 0.71 CTSK (0.48) APLNRCTSKCTSSCTSLCTSB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5563156-A ANTICOAGULANTS, ANTIASTHMA AGENTS MERRELL PHARMACEUTICALS INC. (US) 1996-10-08 US disclosed
US-5498779-A ANTICOAGULANTS AND TREATMENT OF ASTHMA MERRELL PHARMACEUTICALS INC. (US) 1996-03-12 US disclosed
US-5391705-A Anticoagulants, treats thrombophlebitis, coronary thrombosis and asthma MERRELL DOW PHARMACEUTICALS INC. (US) 1995-02-21 US disclosed
EP-0504064-A1 Novel thrombin inhibitors MERRELL PHARMACEUTICALS INC. (US) 1992-09-16 EP disclosed