SCHEMBL8976499

SCHEMBL8976499

COc1ccc(CC(C)(N)c2ccccc2)cc1

nearest known ligand 0.70

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
LTA4H P09960 2/20 0.52
KMT2A Q03164 1/20 0.48
KIF11 P52732 2/20 0.47
KCNH2 Q12809 1/20 0.47
TAAR1 Q96RJ0 2/20 0.46
SLC6A2 P23975 1/20 0.46
CASR P41180 1/20 0.44
SIGMAR1 Q99720 2/20 0.44
CA4 P22748 1/20 0.43
IDO1 P14902 2/20 0.43
AGXT P21549 2/20 0.43
MMP1 P03956 1/20 0.43
MMP13 P45452 1/20 0.43
TDP1 Q9NUW8 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
LMNA P02545 1/20 0.42
HTT P42858 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5305755 0.93 LTA4H (0.52) LTA4HKIF11KCNH2TAAR1SLC6A2
Maleic Acid SCHEMBL8867414 0.89 ALDH1A1 (0.48) KMT2AKIF11TAAR1MMP1MMP13
Fumaric Acid SCHEMBL8867443 0.89 ALDH1A1 (0.48) KMT2AKIF11TAAR1MMP1MMP13
SCHEMBL17964411 0.86 LTA4H (0.55) LTA4HKMT2AKIF11KCNH2TAAR1
SCHEMBL855070 0.83 TAAR1 (0.64) KIF11TAAR1SLC6A2LMNASMN1; SMN2
Fumaric Acid SCHEMBL8866060 0.82 MMP1 (0.47) KMT2AKIF11TAAR1SLC6A2MMP1
Maleic Acid SCHEMBL8866047 0.82 MMP1 (0.47) KMT2AKIF11TAAR1SLC6A2MMP1
SCHEMBL2671508 0.82 LTA4H (0.60) LTA4HKMT2ATAAR1SLC6A2CASR
SCHEMBL5308325 0.82 KIF11 (0.50) KIF11TAAR1SLC6A2CASRSIGMAR1
SCHEMBL8865724 0.82 MAOB (0.57) LTA4HSLC6A2L3MBTL1LMNASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5539120-A Arylalkyl-amines having anticonvulsant and neuroprotective properties AGENCE SPATIALE EUROPEENNE (FR) 1996-07-23 US claimed
EP-0356035-B1 Arylkalkyl-amines and -amides having anticonvulsant and neuroprotective properties ASTRA AB (SE) 1996-03-13 EP claimed
WO-1991011995-A1 ARYLALKYL-AMINES AND -AMIDES HAVING ANTICONVULSANT AND NEUROPROTECTIVE PROPERTIES FISONS CORPORATION (US) 1991-08-22 WO claimed
EP-0356035-A2 Arylkalkyl-amines and -amides having anticonvulsant and neuroprotective properties Astra Aktiebolag (SE) 1990-02-28 EP claimed