SCHEMBL8976527

SCHEMBL8976527

CN(C)c1ccc2[nH]cnc(=O)c2c1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IP6K1 Q92551 3/20 0.58
KDM4E B2RXH2 5/20 0.46
AR P10275 2/20 0.43
PDE3B Q13370 1/20 0.42
PDE3A Q14432 1/20 0.42
MEN1 O00255 1/20 0.40
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
KMT2A Q03164 1/20 0.40
ALDH1A1 P00352 5/20 0.38
ELANE P08246 3/20 0.37
HSD17B10 Q99714 3/20 0.36
GAA P10253 2/20 0.36
USP2 O75604 1/20 0.36
PKM P14618 1/20 0.36
CASP1 P29466 1/20 0.36
CASP7 P55210 1/20 0.36
QPCT Q16769 1/20 0.36
MAPT P10636 2/20 0.36
POLB P06746 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1507612 0.77 PARP1 (0.54) KDM4EMEN1NPC1RAB9AKMT2A
SCHEMBL1584889 0.75 PIM1 (0.56) MEN1KMT2AALDH1A1MAPTHPGD
SCHEMBL3795673 0.75 IP6K1 (0.56) IP6K1KDM4EMEN1NPC1RAB9A
SCHEMBL31361978 0.75 IP6K1 (0.56) IP6K1KDM4EMEN1NPC1RAB9A
SCHEMBL8622177 0.75 ACVR1 (0.46) IP6K1PDE3BPDE3AMEN1NPC1
SCHEMBL2191063 0.74 PARP1 (0.54) KDM4EKMT2AALDH1A1GAAGLA
SCHEMBL2191001 0.74 PARP1 (0.54) ALDH1A1GAAHPGD
SCHEMBL216175 0.74 PARP1 (0.54) MEN1KMT2AALDH1A1QPCTMAPT
SCHEMBL8700858 0.74 PARP1 (0.54) KDM4EARNPC1RAB9AALDH1A1
SCHEMBL2574527 0.74 LMNA (0.57) KDM4EMEN1KMT2AALDH1A1HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5580870-A ANTICARCINOGENIC AGENTS ZENECA LIMITED (GB) 1996-12-03 US disclosed
EP-0602851-B1 Quinazoline derivatives ZENECA LTD (GB) 1996-10-09 EP disclosed
EP-0602851-A1 Quinazoline derivatives ZENECA LIMITED (GB) 1994-06-22 EP disclosed