SCHEMBL8978266

SCHEMBL8978266

CCOC(=O)CC(=O)CCCc1c[nH]c2ccccc12

nearest known ligand 0.81

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.81
CYP1A2 P05177 1/20 0.81
CYP3A4 P08684 1/20 0.81
CYP2D6 P10635 1/20 0.81
CYP2C9 P11712 1/20 0.81
CYP2C19 P33261 1/20 0.81
PKM P14618 1/20 0.64
ALDH1A1 P00352 7/20 0.62
KDM4E B2RXH2 3/20 0.58
L3MBTL1 Q9Y468 1/20 0.58
NPC1 O15118 1/20 0.58
MAPT P10636 6/20 0.58
MEN1 O00255 4/20 0.58
KMT2A Q03164 4/20 0.58
HCRTR1 O43613 1/20 0.56
HPGD P15428 2/20 0.55
TSHR P16473 1/20 0.55
TDP1 Q9NUW8 1/20 0.55
MTNR1A P48039 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9374131 0.90 SMN1; SMN2 (1.00) SMN1; SMN2CYP1A2CYP3A4CYP2D6CYP2C9
Hydrochloric Acid SCHEMBL9368572 0.89 SMN1; SMN2 (0.97) SMN1; SMN2CYP1A2CYP3A4CYP2D6CYP2C9
Hydrochloric Acid SCHEMBL9369222 0.89 SMN1; SMN2 (0.97) SMN1; SMN2CYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL7399266 0.86 SMN1; SMN2 (0.92) SMN1; SMN2CYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL8366567 0.85 PKM (0.80) SMN1; SMN2CYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL392573 0.84 SMN1; SMN2 (0.85) SMN1; SMN2CYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL10031581 0.83 ALDH1A1 (0.69) SMN1; SMN2CYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL1358575 0.82 CYP1A2 (0.76) SMN1; SMN2CYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL7397625 0.81 CYP1A2 (0.73) SMN1; SMN2CYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL17396906 0.79 SMN1; SMN2 (0.67) SMN1; SMN2CYP1A2CYP3A4CYP2D6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5484940-A ULTRAVIOLET RADIATION ABSORBERS FOR PLASTICS, AMYLOID PEPTIDE INHIBITORS, ALZHEIMER*S DISEASE ATHENA NEUROSCIENCES, INC. 1996-01-16 US disclosed