SCHEMBL8980204

SCHEMBL8980204

Nc1ccc2[nH]c(-c3ccccc3)cc(=O)c2c1

nearest known ligand 0.73

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE10A Q9Y233 2/20 0.73
HPGD P15428 7/20 0.68
LMNA P02545 6/20 0.68
ALDH1A1 P00352 5/20 0.68
KDM4E B2RXH2 4/20 0.68
TP53 P04637 2/20 0.68
HSD17B10 Q99714 2/20 0.68
NPC1 O15118 2/20 0.68
RAB9A P51151 2/20 0.68
SMN1; SMN2 Q16637 2/20 0.68
MEN1 O00255 2/20 0.68
KMT2A Q03164 2/20 0.68
TUBB4A P04350 2/20 0.68
TUBB P07437 2/20 0.68
TUBA3C P0DPH7 2/20 0.68
TUBA1B P68363 2/20 0.68
TUBA4A P68366 2/20 0.68
TUBB4B P68371 2/20 0.68
TUBB3 Q13509 2/20 0.68
TUBB2A Q13885 2/20 0.68

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8980201 0.84 PDE10A (0.72) PDE10AHPGDLMNAALDH1A1KDM4E
SCHEMBL2630603 0.83 HPGD (0.76) PDE10AHPGDLMNAALDH1A1KDM4E
SCHEMBL29411863 0.81 HPGD (1.00) PDE10AHPGDLMNAALDH1A1KDM4E
SCHEMBL367268 0.81 HPGD (1.00) PDE10AHPGDLMNAALDH1A1KDM4E
SCHEMBL9385766 0.81 HPGD (0.68) PDE10AHPGDLMNAALDH1A1KDM4E
SCHEMBL2799465 0.81 HPGD (1.00) PDE10AHPGDLMNAALDH1A1KDM4E
SCHEMBL6534299 0.81 HPGD (1.00) HPGDLMNAALDH1A1KDM4ETP53
SCHEMBL30935740 0.81 KMT2A (1.00) PDE10AHPGDLMNAALDH1A1KDM4E
SCHEMBL1273139 0.81 HPGD (0.68) PDE10AHPGDLMNAALDH1A1KDM4E
SCHEMBL8980401 0.81 ALDH1A1 (0.66) HPGDLMNAALDH1A1KDM4ENPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5571822-A AMINO-2-PHENYL-4-QUINOLONE DERIVATIVES THE UNIVERSITY OF NORTH CAROLINA AT CHAPEL HILL (US) 1996-11-05 US disclosed
WO-1996010563-A1 2-ARYL-4-QUINOLONES AS ANTITUMOR COMPOUNDS THE UNIVERSITY OF NORTH CAROLINA AT CHAPEL HILL (US) 1996-04-11 WO disclosed