SCHEMBL8980495

SCHEMBL8980495

O=C1Cc2ccccc2N=C1c1ccccc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 1/20 0.42
MAPT P10636 6/20 0.41
LMNA P02545 3/20 0.41
GAA P10253 2/20 0.41
RARA P10276 1/20 0.41
RARB P10826 1/20 0.41
RXRA P19793 1/20 0.41
RXRB P28702 1/20 0.41
RXRG P48443 1/20 0.41
NOS3 P29474 1/20 0.40
NOS1 P29475 1/20 0.40
NOS2 P35228 1/20 0.40
ALDH1A1 P00352 6/20 0.39
SIGMAR1 Q99720 1/20 0.39
BCHE P06276 1/20 0.38
CES1 P23141 1/20 0.38
CFTR P13569 1/20 0.36
GOPC Q9HD26 1/20 0.36
KDM4E B2RXH2 3/20 0.36
NPC1 O15118 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14507199 0.78 IDO1 (0.50) IDO1MAPTLMNAGAARARA
SCHEMBL28634257 0.77 LMNA (0.39) MAPTLMNAGAABCHEKMT2A
SCHEMBL3443792 0.76 KDM4E (0.41) MAPTLMNANOS3NOS1NOS2
SCHEMBL15066599 0.76 BCHE (0.42) MAPTLMNARARARARBRXRA
SCHEMBL16243903 0.75 MEN1 (0.40) MAPTLMNARARARARBRXRA
SCHEMBL3626217 0.73 NOS3 (0.52) MAPTNOS3NOS1NOS2ALDH1A1
SCHEMBL9674946 0.73 NOS3 (0.42) MAPTLMNANOS3NOS1NOS2
SCHEMBL8177168 0.73 NOS3 (0.42) MAPTLMNAGAANOS3NOS1
SCHEMBL4145325 0.73 NOS3 (0.42) MAPTLMNANOS3NOS1NOS2
SCHEMBL2866347 0.73 MAOA (0.45) MAPTRARARARBRXRARXRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103391932-B For suppressing the heterogeneous ring compound of PASK BIOENERGENIX (US) 2015-10-14 CN disclosed
CN-103391932-A Heterocyclic compounds for the inhibition of pask BIOENERGENIX 2013-11-13 CN disclosed
US-5571822-A AMINO-2-PHENYL-4-QUINOLONE DERIVATIVES THE UNIVERSITY OF NORTH CAROLINA AT CHAPEL HILL (US) 1996-11-05 US disclosed
WO-1996010563-A1 2-ARYL-4-QUINOLONES AS ANTITUMOR COMPOUNDS THE UNIVERSITY OF NORTH CAROLINA AT CHAPEL HILL (US) 1996-04-11 WO disclosed