SCHEMBL8983608

SCHEMBL8983608

C[Si](C)(C)C#CCCCS(C)(=O)=O

nearest known ligand 0.38

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
NLRP3 Q96P20 1/20 0.38
ALDH1A1 P00352 1/20 0.35
LMNA P02545 1/20 0.35
TP53 P04637 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8983703 0.79 NLRP3 (0.35) NLRP3ALDH1A1LMNATP53
SCHEMBL16420274 0.75 RAB9A (0.33) LMNA
SCHEMBL31725737 0.73 RAB9A (0.38)
SCHEMBL790554 0.72 KDM4E (0.56) ALDH1A1LMNA
SCHEMBL14480051 0.72
SCHEMBL23014988 0.71 TSHR (0.54) ALDH1A1LMNA
SCHEMBL23014933 0.71 TSHR (0.54) ALDH1A1LMNA
SCHEMBL23532681 0.69
SCHEMBL588584 0.69 TSHR (0.39) ALDH1A1LMNA
SCHEMBL11651534 0.69

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5550239-A REACTING TRIALKYLSILYL N-PENTYLPIPERAZINYLPYRIMIDINE DERIVATIVE WITH 4-AMINO-3-IODO-BENZENESULFONAMIDE COMPOUND IN PALLADIUM CATALYZED HETEROANNULATION STEP, REMOVING TRIALKYLSILYL GROUP WITH MINERAL ACID, BASIFYING BRISTOL-MYERS SQUIBB COMPANY (US) 1996-08-27 US disclosed
EP-0711769-A1 Improved process for large-scale production of BMS 180048 and analogs BRISTOL-MYERS SQUIBB COMPANY (US) 1996-05-15 EP disclosed