SCHEMBL8985488

SCHEMBL8985488

CNC(=O)c1cc(-c2ccc(SC)cc2)c(-c2ccc(Cl)cc2)s1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.55
CYP1A2 P05177 1/20 0.55
POLB P06746 1/20 0.55
CYP2D6 P10635 1/20 0.55
CYP2C9 P11712 1/20 0.55
CYP2C19 P33261 1/20 0.55
SMN1; SMN2 Q16637 3/20 0.45
GAA P10253 3/20 0.45
LMNA P02545 2/20 0.45
MAPT P10636 4/20 0.45
KDM4E B2RXH2 3/20 0.45
HPGD P15428 1/20 0.45
HTT P42858 1/20 0.45
HSD17B10 Q99714 1/20 0.45
NPSR1 Q6W5P4 2/20 0.44
RXFP1 Q9HBX9 1/20 0.44
PLK1 P53350 2/20 0.43
OPRD1 P41143 1/20 0.43
RAB9A P51151 3/20 0.40
KMT2A Q03164 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8985429 0.94 KDM4E (0.50) ALDH1A1CYP1A2POLBCYP2D6CYP2C9
SCHEMBL8985425 0.88 MAPK14 (0.52) ALDH1A1CYP1A2POLBCYP2D6CYP2C9
SCHEMBL8985326 0.88 MAPK14 (0.52) ALDH1A1CYP1A2POLBCYP2D6CYP2C9
SCHEMBL8985419 0.86 MAPK14 (0.52) ALDH1A1CYP1A2POLBCYP2D6CYP2C9
SCHEMBL8985259 0.86 MAPK14 (0.50) ALDH1A1CYP1A2POLBCYP2D6CYP2C9
SCHEMBL8985238 0.85 OPRD1 (0.63) ALDH1A1CYP1A2POLBCYP2D6CYP2C9
SCHEMBL8985209 0.82 SMN1; SMN2 (0.45) ALDH1A1CYP1A2POLBCYP2D6CYP2C9
SCHEMBL8985220 0.81 PTGS2 (0.49) ALDH1A1CYP1A2POLBCYP2D6CYP2C9
SCHEMBL8985541 0.78 MAPK14 (0.56) ALDH1A1LMNAKDM4EHPGDOPRD1
SCHEMBL8985191 0.77 MAPK14 (0.60) ALDH1A1CYP1A2CYP2C9CYP2C19SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5571810-A ANTIINFLAMMATORY AGENTS, ANALGESICS, COLLAGEN DISEASES FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1996-11-05 US disclosed
EP-0593761-A1 NEW THIOPHENE DERIVATIVES FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1994-04-27 EP disclosed
WO-1991019708-A1 NEW THIOPHENE DERIVATIVES FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1991-12-26 WO disclosed