SCHEMBL8985491

SCHEMBL8985491

CSc1ccc(-c2cc(Br)sc2-c2ccc(NCC=O)cc2)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 4/20 0.43
CYP1A2 P05177 4/20 0.43
CYP2C9 P11712 4/20 0.43
CYP2C19 P33261 4/20 0.43
PTGS1 P23219 3/20 0.43
CYP3A4 P08684 3/20 0.43
KDM4E B2RXH2 2/20 0.43
MT-CO1 P00395 1/20 0.43
MT-CO2 P00403 1/20 0.43
HPGD P15428 1/20 0.43
TSHR P16473 1/20 0.43
HSD17B10 Q99714 1/20 0.43
RAB9A P51151 3/20 0.34
NPC1 O15118 3/20 0.34
MAPT P10636 3/20 0.34
CYP2D6 P10635 1/20 0.34
MEN1 O00255 4/20 0.33
KMT2A Q03164 4/20 0.33
RECQL P46063 1/20 0.33
ALDH1A1 P00352 3/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8985459 0.87 CYP1A2 (0.37) PTGS2CYP1A2CYP2C9CYP2C19PTGS1
SCHEMBL8985514 0.85 PTGS2 (0.42) PTGS2CYP1A2CYP2C9CYP2C19PTGS1
SCHEMBL8985336 0.84 MAPK14 (0.45) PTGS2PTGS1KDM4ERAB9ANPC1
SCHEMBL8985319 0.84 PTGS2 (0.34) PTGS2CYP1A2CYP2C9CYP2C19PTGS1
SCHEMBL8985260 0.83 PTGS2 (0.65) PTGS2CYP1A2CYP2C9CYP2C19PTGS1
SCHEMBL8985448 0.83 OPRD1 (0.39) PTGS2PTGS1KDM4ERAB9ANPC1
SCHEMBL8985328 0.82 PTGS1 (0.43) PTGS2CYP1A2CYP2C9CYP2C19PTGS1
SCHEMBL8985524 0.80 MAPK14 (0.51) PTGS2PTGS1KDM4EHPGDTSHR
SCHEMBL24035226 0.78 MEN1 (0.49) CYP1A2CYP2C9CYP2C19CYP3A4KDM4E
SCHEMBL8985493 0.77 PTGS1 (0.41) PTGS2CYP1A2CYP2C9CYP2C19PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5571810-A ANTIINFLAMMATORY AGENTS, ANALGESICS, COLLAGEN DISEASES FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1996-11-05 US disclosed
EP-0593761-A1 NEW THIOPHENE DERIVATIVES FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1994-04-27 EP disclosed