SCHEMBL8987649

SCHEMBL8987649

COc1ccc(CN(CCCC(N)=O)Cc2ccc(OC)cc2)cc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEP1B Q16820 2/20 0.55
ACHE P22303 2/20 0.50
NR1H3 Q13133 2/20 0.50
BCHE P06276 1/20 0.50
ALOX5 P09917 2/20 0.48
ALDH1A1 P00352 1/20 0.48
HTT P42858 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.48
F2RL1 P55085 1/20 0.45
APLNR P35414 1/20 0.45
TDP1 Q9NUW8 1/20 0.45
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
PTPN1 P18031 1/20 0.44
USP2 O75604 1/20 0.44
TSHR P16473 1/20 0.44
TSPO P30536 1/20 0.43
BMP1 P13497 1/20 0.43
CA1 P00915 1/20 0.43
CA2 P00918 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9172532 0.88 MEP1B (0.58) MEP1BACHENR1H3BCHEALOX5
SCHEMBL9540871 0.83 ACHE (0.56) MEP1BACHENR1H3BCHEALOX5
SCHEMBL8987663 0.82 HDAC3 (0.43) MEP1BACHEBCHEALDH1A1
SCHEMBL27200631 0.81 MEP1B (0.60) MEP1BACHEBCHEALDH1A1HTT
SCHEMBL23857640 0.79 MEP1B (0.58) MEP1BACHEBCHEALOX5ALDH1A1
SCHEMBL23857357 0.79 MEP1B (0.58) MEP1BACHEBCHEALDH1A1HTT
SCHEMBL8987627 0.79 CYP2C9 (0.47) ALDH1A1HTT
SCHEMBL14066026 0.79 ACHE (0.51) MEP1BACHENR1H3BCHETDP1
SCHEMBL8987514 0.78 HDAC3 (0.61) ACHEBCHEALOX5CA1CA2
SCHEMBL659052 0.78 ALOX5 (0.68) ALOX5ALDH1A1F2RL1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0345068-B1 Agonist of gamma-aminobutyric acid WYETH JOHN & BROTHER LTD (GB) 1995-03-15 EP claimed
US-5527955-A AGONIST OF GAMMA AMINOBUTYRIC ACID JOHN WYETH & BROTHER, LIMITED (GB) 1996-06-18 US disclosed
EP-0345068-B1 Agonist of gamma-aminobutyric acid WYETH JOHN & BROTHER LTD (GB) 1995-03-15 EP disclosed
EP-0345068-A2 Agonist of gamma-aminobutyric acid JOHN WYETH & BROTHER LIMITED (GB) 1989-12-06 EP disclosed