SCHEMBL8987663

SCHEMBL8987663

Cc1ccc(CN(CCCC(N)=O)Cc2ccc(C)cc2)cc1

nearest known ligand 0.44

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 2/20 0.43
HDAC1 Q13547 2/20 0.43
HDAC2 Q92769 2/20 0.43
HDAC8 Q9BY41 2/20 0.43
NCOR2 Q9Y618 2/20 0.43
MAPT P10636 1/20 0.42
RORC P51449 1/20 0.40
SLC1A5 Q15758 1/20 0.40
ALDH1A1 P00352 1/20 0.39
HSP90AA1 P07900 1/20 0.38
BCHE P06276 1/20 0.38
ACHE P22303 1/20 0.38
MEP1B Q16820 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8987683 0.86 HDAC3 (0.46) HDAC3HDAC1HDAC2HDAC8NCOR2
SCHEMBL8987627 0.83 CYP2C9 (0.47) HDAC3HDAC1HDAC2HDAC8NCOR2
SCHEMBL8987514 0.82 HDAC3 (0.61) HDAC3HDAC1HDAC2HDAC8NCOR2
SCHEMBL8987649 0.82 MEP1B (0.55) ALDH1A1BCHEACHEMEP1B
Hydrochloric Acid SCHEMBL9132070 0.81 HDAC3 (0.59) HDAC3HDAC1HDAC2HDAC8NCOR2
P-Xylene SCHEMBL746836 0.77 ALDH1A1 (0.52) HDAC3HDAC1HDAC2HDAC8NCOR2
SCHEMBL661277 0.76 PLAAT3 (0.51) HDAC3HDAC1HDAC2HDAC8
P-Xylene SCHEMBL6033011 0.75 ALDH1A1 (0.50) HDAC3HDAC1HDAC2HDAC8NCOR2
P-Xylene SCHEMBL18427877 0.75 ALDH1A1 (0.50) HDAC3HDAC1HDAC2HDAC8NCOR2
SCHEMBL4367534 0.74 TDP1 (0.50) HDAC3HDAC1HDAC2HDAC8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0345068-B1 Agonist of gamma-aminobutyric acid WYETH JOHN & BROTHER LTD (GB) 1995-03-15 EP claimed
EP-0345068-A2 Agonist of gamma-aminobutyric acid JOHN WYETH & BROTHER LIMITED (GB) 1989-12-06 EP claimed
US-5527955-A AGONIST OF GAMMA AMINOBUTYRIC ACID JOHN WYETH & BROTHER, LIMITED (GB) 1996-06-18 US disclosed
EP-0345068-B1 Agonist of gamma-aminobutyric acid WYETH JOHN & BROTHER LTD (GB) 1995-03-15 EP disclosed
US-5321047-A Antidepressant JOHN WYETH & BROTHER, LIMITED (GB) 1994-06-14 US disclosed
EP-0345068-A2 Agonist of gamma-aminobutyric acid JOHN WYETH & BROTHER LIMITED (GB) 1989-12-06 EP disclosed