SCHEMBL8987668

SCHEMBL8987668

N#CCCCN(Cc1ccccc1)C(c1ccccc1)c1ccccc1

nearest known ligand 0.44

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
OPRD1 P41143 1/20 0.44
SIGMAR1 Q99720 1/20 0.42
ALDH1A1 P00352 6/20 0.42
GAA P10253 2/20 0.40
POLB P06746 2/20 0.40
KMT2A Q03164 2/20 0.40
TSHR P16473 1/20 0.40
NPBWR1 P48145 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
MCHR1 Q99705 1/20 0.40
KCNN4 O15554 1/20 0.36
KCNA5 P22460 1/20 0.36
KDM4E B2RXH2 1/20 0.36
LMNA P02545 1/20 0.36
AR P10275 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
MEN1 O00255 1/20 0.34
MAOB P27338 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL154270 0.81 ALDH1A1 (0.48) ALDH1A1GAAPOLBKMT2AKCNN4
SCHEMBL7877735 0.81 ALDH1A1 (0.48) OPRD1ALDH1A1GAAPOLBKCNN4
Hydrochloric Acid SCHEMBL11203276 0.80 ALDH1A1 (0.47) OPRD1ALDH1A1GAAPOLBKCNN4
SCHEMBL10962715 0.78 POLB (0.47) ALDH1A1GAAPOLBAR
SCHEMBL8987693 0.76 OPRD1 (0.52) OPRD1SIGMAR1
SCHEMBL7982573 0.76 ALDH1A1 (0.53) OPRD1SIGMAR1ALDH1A1GAAKMT2A
SCHEMBL8987713 0.76 HDAC3 (0.49) ALDH1A1GAAPOLBMAOB
SCHEMBL17508109 0.76 ALDH1A1 (0.47) OPRD1ALDH1A1GAAPOLBMAOB
SCHEMBL154265 0.75 KCNH2 (0.51) SIGMAR1KDM4EMAOB
SCHEMBL149999 0.75 SIGMAR1 (0.59) SIGMAR1ALDH1A1TSHRLMNAMAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5527955-A AGONIST OF GAMMA AMINOBUTYRIC ACID JOHN WYETH & BROTHER, LIMITED (GB) 1996-06-18 US disclosed
EP-0345068-B1 Agonist of gamma-aminobutyric acid WYETH JOHN & BROTHER LTD (GB) 1995-03-15 EP disclosed
US-5321047-A Antidepressant JOHN WYETH & BROTHER, LIMITED (GB) 1994-06-14 US disclosed
EP-0345068-A2 Agonist of gamma-aminobutyric acid JOHN WYETH & BROTHER LIMITED (GB) 1989-12-06 EP disclosed