SCHEMBL8988701

SCHEMBL8988701

COC(=O)CCc1ccc(C2=C(OC)CN(c3ccc4c(c3)CCC4N)C2=O)cc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 2/20 0.38
HDAC1 Q13547 1/20 0.35
CTSD P07339 1/20 0.34
PTPN1 P18031 1/20 0.33
F10 P00742 1/20 0.33
GCK P35557 2/20 0.32
LIPG Q9Y5X9 1/20 0.31
GHSR Q92847 1/20 0.31
EP300 Q09472 1/20 0.31
ACHE P22303 1/20 0.31
TBXA2R P21731 1/20 0.31
PTGER4 P35408 1/20 0.31
MCHR1 Q99705 1/20 0.30
KDM4E B2RXH2 1/20 0.30
USP2 O75604 1/20 0.30
CYP3A4 P08684 1/20 0.30
HIF1A Q16665 1/20 0.30
TDP1 Q9NUW8 1/20 0.30
MMP2 P08253 1/20 0.30
ANPEP P15144 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8988899 0.95 HRH3 (0.38) HRH3HDAC1CTSDPTPN1MCHR1
Hydrochloric Acid SCHEMBL8988652 0.91 HRH3 (0.33) HRH3F10GCKEP300
Hydrochloric Acid SCHEMBL8988625 0.86 OPRD1 (0.36) HRH3MCHR1
SCHEMBL8988799 0.82 HRH3 (0.40) HRH3HDAC1CTSDPTPN1KDM4E
SCHEMBL7384118 0.82 HRH3 (0.40) HRH3HDAC1CTSDF10ACHE
Hydrochloric Acid SCHEMBL8988618 0.81 HRH3 (0.39) HRH3HDAC1CTSDPTPN1KDM4E
Hydrochloric Acid SCHEMBL7281181 0.81 HRH3 (0.39) HRH3HDAC1CTSDF10ACHE
SCHEMBL8988630 0.79 PTPN1 (0.40) HRH3HDAC1CTSDPTPN1
SCHEMBL8988853 0.77 HRH3 (0.37) HRH3HDAC1CTSDPTPN1F10
SCHEMBL8988689 0.77 ITGB3 (0.43) HRH3HDAC1PTPN1F10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5489693-A ANTICOAGULANTS DR. KARK THOMAE, GMBH (DE) 1996-02-06 US disclosed
EP-0567968-A1 Cyclic imino derivatives, medicaments containing these compounds and processes for the production thereof Dr. Karl Thomae GmbH (DE) 1993-11-03 EP disclosed