SCHEMBL8989237

SCHEMBL8989237

Cc1cnc(-c2ccc(C(F)(F)F)cc2)n1C

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 5/20 0.47
TP53 P04637 2/20 0.47
GAA P10253 2/20 0.47
MAPT P10636 2/20 0.47
POLB P06746 1/20 0.47
SIGMAR1 Q99720 1/20 0.43
KDM4E B2RXH2 2/20 0.41
ALDH1A1 P00352 1/20 0.41
LMNA P02545 1/20 0.41
CYP1A2 P05177 1/20 0.41
HPGD P15428 1/20 0.41
NFKB1 P19838 1/20 0.41
BLM P54132 1/20 0.41
PMP22 Q01453 1/20 0.41
HSD17B10 Q99714 1/20 0.41
PPARD Q03181 2/20 0.40
TDP2 O95551 1/20 0.40
HSD11B1 P28845 1/20 0.39
COMT P21964 1/20 0.39
DYRK3 O43781 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24173752 0.84 ALDH1A1 (0.50) KIF11POLBSIGMAR1KDM4EALDH1A1
SCHEMBL3534328 0.83 TP53 (0.45) KIF11TP53GAAMAPTPOLB
SCHEMBL8989158 0.78 PPARD (0.47) KIF11TP53GAAMAPTPOLB
SCHEMBL8989180 0.78 PPARD (0.40) KIF11TP53GAAMAPTPOLB
SCHEMBL15167073 0.78 MEN1 (0.46) TP53GAAMAPTPOLBSIGMAR1
SCHEMBL12759486 0.77 TP53 (0.46) TP53GAAMAPTPOLBHSD11B1
SCHEMBL8989228 0.76 MAP4K4 (0.53) TP53MAPTALDH1A1CYP1A2HSD11B1
SCHEMBL8453399 0.75 HPGDS (0.58) GAAMAPTKDM4EALDH1A1CYP1A2
SCHEMBL15168293 0.75 SMN1; SMN2 (0.44) TP53GAAMAPTPOLBKDM4E
SCHEMBL11624181 0.74 KIF11 (0.41) KIF11TP53GAAMAPTPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5545645-A Heterocyclic derivatives in the treatment of ischaemia and related diseases SYNTEX PHARMACEUTICALS, LIMITED (GB) 1996-08-13 US disclosed
US-5428037-A Piperazine derivatives; calcium and sodium channel antagonists SYNTEX PHARMACEUTICALS, LTD. (GB) 1995-06-27 US disclosed