SCHEMBL8989727

SCHEMBL8989727

Nc1cc(CCc2ccccc2)ccn1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOS3 P29474 3/20 0.57
NOS1 P29475 3/20 0.57
NOS2 P35228 3/20 0.57
GABRP O00591 2/20 0.55
GABRD O14764 2/20 0.55
GABRA1 P14867 2/20 0.55
GABRB1 P18505 2/20 0.55
GABRG2 P18507 2/20 0.55
GABRB3 P28472 2/20 0.55
GABRA5 P31644 2/20 0.55
GABRA3 P34903 2/20 0.55
GABRA2 P47869 2/20 0.55
GABRB2 P47870 2/20 0.55
GABRA4 P48169 2/20 0.55
GABRE P78334 2/20 0.55
GABRA6 Q16445 2/20 0.55
GABRG1 Q8N1C3 2/20 0.55
GABRG3 Q99928 2/20 0.55
GABRQ Q9UN88 2/20 0.55
MAOA P21397 4/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1600990 0.84 NOS3 (0.57) NOS3NOS1NOS2GABRPGABRD
SCHEMBL4134209 0.79 NOS3 (0.61) NOS3NOS1NOS2GABRPGABRD
SCHEMBL16502197 0.79 NR3C2 (0.51) MAOAMAOBNR3C2KDM4ESMN1; SMN2
SCHEMBL4543342 0.79 NR3C2 (0.59) NOS3NOS1NOS2GABRPGABRD
SCHEMBL23706252 0.78 NR3C2 (0.51) MAOAMAOBNR3C2CYP2A6HTR2A
SCHEMBL18476749 0.78 NOS3 (0.59) NOS3NOS1NOS2GABRPGABRD
SCHEMBL318128 0.78 NOS3 (0.59) NOS3NOS1NOS2GABRPGABRD
Hydrochloric Acid SCHEMBL29481452 0.78 NOS3 (0.59) NOS3NOS1NOS2GABRPGABRD
SCHEMBL105611 0.78 NOS2 (0.70) NOS3NOS1NOS2GABRPGABRD
Hydrochloric Acid SCHEMBL6953232 0.78 NOS3 (0.59) NOS3NOS1NOS2GABRPGABRD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5527796-A ANALGESICS, ANTIINFLAMMATORY AGENTS CHEMISCH PHARMAZEUTISCHE FORSCHUNGSGESELLSCHAFT M.B.H. (AT) 1996-06-18 US disclosed
EP-0576906-A1 Thienothiazine derivatives, process for their preparation and their use as antiinflammatory and analgesic agents Chemisch Pharmazeutische Forschungsgesellschaft m.b.H. (AT) 1994-01-05 EP disclosed