SCHEMBL8989833

SCHEMBL8989833

O=C(O)Cc1ccc(Br)c(C2CCCCC2N2CCOCC2)c1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 7/20 0.38
THRA P10827 2/20 0.38
THRB P10828 2/20 0.38
KCNA5 P22460 1/20 0.37
SCN5A Q14524 1/20 0.37
OPRK1 P41145 4/20 0.36
OPRM1 P35372 2/20 0.36
TP53 P04637 2/20 0.36
CYP3A4 P08684 2/20 0.36
CYP2D6 P10635 2/20 0.36
TSHR P16473 2/20 0.36
KMT2A Q03164 2/20 0.36
ALDH1A1 P00352 2/20 0.36
MEN1 O00255 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP2C19 P33261 1/20 0.36
MTOR P42345 1/20 0.36
RAB9A P51151 1/20 0.36
OPRD1 P41143 1/20 0.36
MAPK8 P45983 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8989860 0.80 KCNA5 (0.39) SIGMAR1THRBKCNA5SCN5AOPRK1
SCHEMBL7799100 0.76 KCNA5 (0.41) SIGMAR1KCNA5SCN5ACYP3A4TSHR
Hydrochloric Acid SCHEMBL7803104 0.75 KCNA5 (0.40) SIGMAR1KCNA5SCN5ACYP3A4TSHR
SCHEMBL8989847 0.70 OPRM1 (0.43) OPRK1OPRM1
SCHEMBL7799090 0.69 OPRM1 (0.40) SIGMAR1KCNA5SCN5AOPRK1OPRM1
SCHEMBL8989835 0.69 UTS2R (0.47) OPRK1OPRM1HRH3
Hydrochloric Acid SCHEMBL8989821 0.68 UTS2R (0.47) OPRK1OPRM1
Hydrochloric Acid SCHEMBL7798770 0.68 OPRM1 (0.41) KCNA5SCN5AOPRK1OPRM1
SCHEMBL7799084 0.67 OPRM1 (0.40) SIGMAR1KCNA5SCN5AOPRK1OPRM1
SCHEMBL7800794 0.67 HTR7 (0.39) SIGMAR1KCNA5SCN5AOPRK1OPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0720605-A1 AMINOCYCLOHEXYLESTERS AND USES THEREOF UNIVERSITY OF BRITISH COLUMBIA (CA) 1996-07-10 EP claimed
WO-1995008544-A1 AMINOCYCLOHEXYLESTERS AND USES THEREOF THE UNIVERSITY OF BRITISH COLUMBIA (CA) 1995-03-30 WO claimed