SCHEMBL8990028

SCHEMBL8990028

CC(C)CCOC(=O)CBr

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C19 P33261 1/20 0.54
L3MBTL1 Q9Y468 2/20 0.52
ALDH1A1 P00352 3/20 0.50
TRPA1 O75762 2/20 0.50
CYP19A1 P11511 1/20 0.47
CA12 O43570 1/20 0.43
CA1 P00915 1/20 0.43
CA2 P00918 1/20 0.43
CA9 Q16790 1/20 0.43
TDP1 Q9NUW8 2/20 0.42
MAPK1 P28482 2/20 0.39
PKM P14618 2/20 0.39
KDM4E B2RXH2 1/20 0.39
GAA P10253 1/20 0.39
KMT2A Q03164 1/20 0.39
HSD17B10 Q99714 1/20 0.38
EPHX2 P34913 1/20 0.37
ACHE P22303 1/20 0.37
FAAH O00519 1/20 0.36
PPARG P37231 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21883838 0.86 CYP2C19 (0.54) CYP2C19L3MBTL1ALDH1A1TRPA1CYP19A1
SCHEMBL11785901 0.84 FAAH (0.47) CYP2C19L3MBTL1ALDH1A1TRPA1CYP19A1
SCHEMBL2267201 0.81 CYP19A1 (0.50) ALDH1A1CYP19A1CA12CA1CA2
SCHEMBL333015 0.81 ADRA2A (0.50) ALDH1A1CYP19A1CA12CA1CA2
SCHEMBL21883834 0.81 CYP2C19 (0.48) CYP2C19L3MBTL1ALDH1A1TRPA1CYP19A1
SCHEMBL27738473 0.80 TDP1 (0.49) L3MBTL1ALDH1A1CYP19A1CA12CA1
SCHEMBL126952 0.79 NAAA (0.50) ALDH1A1CYP19A1CA12CA1CA2
SCHEMBL901332 0.79 CYP19A1 (0.49) ALDH1A1CYP19A1CA12CA1CA2
SCHEMBL4292777 0.79 CYP19A1 (0.49) ALDH1A1CYP19A1CA12CA1CA2
SCHEMBL2536919 0.79 CYP19A1 (0.49) L3MBTL1ALDH1A1CYP19A1CA12CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11357873-B2 Chiral cyclen compounds and their uses THE HONG KONG POLYTECHNIC UNIVERSITY (CN) 2022-06-14 US disclosed
US-5578633-A VASOPRESSIN AND OXYTOCIN ANTAGONISTS SANOFI (FR) 1996-11-26 US disclosed
US-5481005-A N-sulfonylindoline derivatives, their preparation and the pharmaceutical compositions in which they are present SANOFI (FR) 1996-01-02 US disclosed
US-5397801-A Affinity for vasopressin and ocytocin receptors; disorders of nervous, cardiovascular and gastrointestinal systems SANOFI (FR) 1995-03-14 US disclosed
US-5338755-A Have affinity for vasopressin and ocytocin receptors; intermediates for drugs that act on central nervous system ELF SANOFI (FR) 1994-08-16 US disclosed
US-4563310-A HERBICIDES ZOECON CORPORATION (US) 1986-01-07 US disclosed
EP-0065374-A1 Substituted phosphinates and phosphinothioates and their use for the control of weeds ZOECON CORPORATION (US) 1982-11-24 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11357873-B2 Chiral cyclen compounds and their uses DCTN3, DCTN1, CDK3 CYP2C19 4003/4885L3MBTL1 4523/4885ALDH1A1 3008/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.