SCHEMBL8990561

SCHEMBL8990561

COC(C)(C)C(=O)OCCCl

nearest known ligand 0.33

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ABCB11 O95342 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
TSHR P16473 1/20 0.33
HTR2A P28223 1/20 0.33
PMP22 Q01453 1/20 0.33
PPARA Q07869 1/20 0.33
CYP4F2 P78329 1/20 0.33
CYP4A11 Q02928 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8301609 0.82 ABCB11 (0.34) ABCB11CYP1A2CYP3A4TSHRHTR2A
SCHEMBL6008109 0.80 CYP4F2 (0.41) ABCB11CYP1A2CYP3A4TSHRHTR2A
SCHEMBL23293115 0.80 HCAR2 (0.38) ABCB11CYP1A2CYP3A4TSHRHTR2A
SCHEMBL3910492 0.79 POLB (0.43) CYP1A2CYP3A4CYP4F2CYP4A11
SCHEMBL4675028 0.79 GAA (0.38) ABCB11CYP1A2CYP3A4TSHRHTR2A
SCHEMBL4675025 0.79 ABCB11 (0.31) ABCB11CYP1A2CYP3A4TSHRHTR2A
SCHEMBL7064192 0.78 TDP1 (0.34) ABCB11CYP1A2CYP3A4TSHRHTR2A
SCHEMBL7064188 0.78 ABCB11 (0.30) ABCB11CYP1A2CYP3A4TSHRHTR2A
SCHEMBL9312845 0.77 ALDH1A1 (0.33) TSHR
SCHEMBL11778231 0.77 POLB (0.31)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5587374-A BACTERICIDES TREATING INFECTIONS GLAXO SPA (IT) 1996-12-24 US disclosed
EP-0495953-B1 10-(1-Hydroxyethyl)-11-oxo-1-azatricyclo[7.2.0.0(3,8)]undec-2-ene-2-carboxylic acid esters and a process for preparing thereof GLAXO SPA (IT) 1994-06-08 EP disclosed
EP-0495953-A1 10-(1-Hydoxyethyl)-11-oxo-1-azatricyclo(7.2.0.0(3,8)undec-2-ene-2-carboxylic acid esters and a process for preparing thereof. GLAXO SPA (IT) 1992-07-29 EP disclosed
WO-1992003437-A1 10(1-HYDROXYETHYL)-11-OXO-1-AZATRICYCLO[7.2.0.0.3.8]UNDEC-2-ENE-2-CARBOXYLIC ACID ESTERS AND A PROCESS FOR PREPARING THEREOF GLAXO S.P.A. (IT) 1992-03-05 WO disclosed