SCHEMBL8990709

SCHEMBL8990709

Nc1ncnc(CC(O)c2ccccc2)c1N

nearest known ligand 0.40

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
AOC3 Q16853 5/20 0.40
LMNA P02545 1/20 0.39
KDM4E B2RXH2 2/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
SRC P12931 2/20 0.36
CYP2D6 P10635 1/20 0.36
BCAT2 O15382 1/20 0.36
NPC1 O15118 1/20 0.35
DHFR P00374 1/20 0.35
HPGD P15428 1/20 0.35
AURKA O14965 1/20 0.34
RPS6KB1 P23443 1/20 0.34
RIPK1 Q13546 1/20 0.34
TSHR P16473 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27631895 0.69 DHFR (0.45) AOC3LMNAKDM4EL3MBTL1CYP2D6
SCHEMBL9646578 0.68 AOC3 (0.47) AOC3LMNAKDM4EL3MBTL1BCAT2
SCHEMBL9660286 0.67 LMNA (0.46) AOC3LMNAKDM4EL3MBTL1CYP2D6
SCHEMBL9658892 0.67 LMNA (0.50) AOC3LMNAKDM4EL3MBTL1CYP2D6
SCHEMBL9660899 0.67 LMNA (0.46) AOC3LMNAKDM4EL3MBTL1CYP2D6
SCHEMBL9660894 0.67 LMNA (0.46) AOC3LMNAKDM4EL3MBTL1CYP2D6
SCHEMBL9658896 0.67 LMNA (0.50) AOC3LMNAKDM4EL3MBTL1CYP2D6
SCHEMBL9660282 0.67 LMNA (0.46) AOC3LMNAKDM4EL3MBTL1CYP2D6
SCHEMBL8352649 0.66 SOAT1 (0.53) AOC3LMNAKDM4EL3MBTL1
SCHEMBL2021 0.66 TAAR1 (0.62) AOC3LMNAKDM4EL3MBTL1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5500428-A Furyl-substituted purines and adenosine antagonists IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1996-03-19 US disclosed
US-5300509-A Adenosine antagonists for treating cardiovascular disorders, vasodilation IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1994-04-05 US disclosed
EP-0544445-A2 Furyl-substituted purines, oxazolopyrimidines and pteridines as adenosine antagonists ZENECA LIMITED (GB) 1993-06-02 EP disclosed