SCHEMBL8992699

SCHEMBL8992699

CCCCc1nc(CCN2C(=O)c3ccccc3C2=O)c[nH]1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PKM P14618 1/20 0.49
HSD17B10 Q99714 1/20 0.48
POLB P06746 2/20 0.46
ALDH1A1 P00352 2/20 0.46
MAPT P10636 5/20 0.46
MEN1 O00255 2/20 0.45
KMT2A Q03164 2/20 0.45
ACHE P22303 1/20 0.45
SMN1; SMN2 Q16637 2/20 0.44
LMNA P02545 1/20 0.44
TLR8 Q9NR97 1/20 0.44
TLR7 Q9NYK1 1/20 0.44
NPC1 O15118 1/20 0.44
GAA P10253 1/20 0.44
RAB9A P51151 1/20 0.44
TDP1 Q9NUW8 1/20 0.42
TSHR P16473 1/20 0.42
PDE10A Q9Y233 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP2D6 P10635 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8992759 0.92 PKM (0.51) PKMHSD17B10POLBALDH1A1MAPT
SCHEMBL9052259 0.88 PKM (0.52) PKMHSD17B10POLBALDH1A1MAPT
SCHEMBL7743461 0.80 MAPT (0.58) PKMHSD17B10POLBALDH1A1MAPT
SCHEMBL9372170 0.77 MAPT (0.51) PKMMAPTMEN1KMT2ASMN1; SMN2
SCHEMBL3840247 0.75 HRH3 (0.42) PKMALDH1A1
Biphenyl SCHEMBL7417032 0.75 PARP1 (0.43)
SCHEMBL3841613 0.74 HRH3 (0.41) PKMALDH1A1
Hydrochloric Acid SCHEMBL28183399 0.74 HRH3 (0.41) PKMALDH1A1
SCHEMBL29511230 0.72 CHRM2 (0.61) ALDH1A1MEN1KMT2ATDP1CYP1A2
SCHEMBL149620 0.72 CHRM2 (0.61) ALDH1A1MEN1KMT2ATDP1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5510354-A HYPOTENSIVE AGENTS TANABE SEIYAKU CO., LTD. (JP) 1996-04-23 US disclosed
US-5424316-A Imidazopyridine derivatives for the treatment of hypertension TANABE SEIYAKU CO., LTD. (JP) 1995-06-13 US disclosed
US-5409936-A Useful in prophylaxix; exhibits potent angiotensin ii inhibitory acivities TANABE SEIYAKU CO., LTD. (JP) 1995-04-25 US disclosed
EP-0531874-A1 Imidazopyridine derivatives and process for preparation thereof TANABE SEIYAKU CO., LTD. (JP) 1993-03-17 EP disclosed