SCHEMBL8992759

SCHEMBL8992759

CCCc1nc(CCN2C(=O)c3ccccc3C2=O)c[nH]1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PKM P14618 1/20 0.51
HSD17B10 Q99714 1/20 0.50
ALDH1A1 P00352 4/20 0.48
POLB P06746 2/20 0.48
MAPT P10636 4/20 0.48
MEN1 O00255 2/20 0.47
KMT2A Q03164 2/20 0.47
LMNA P02545 2/20 0.46
SMN1; SMN2 Q16637 2/20 0.46
GAA P10253 2/20 0.46
NPC1 O15118 1/20 0.46
RAB9A P51151 1/20 0.46
TSHR P16473 1/20 0.44
PDE10A Q9Y233 1/20 0.43
GLS O94925 1/20 0.43
CYP1A2 P05177 1/20 0.43
CYP2D6 P10635 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
HPGD P15428 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8992699 0.92 PKM (0.49) PKMHSD17B10ALDH1A1POLBMAPT
SCHEMBL9052259 0.90 PKM (0.52) PKMHSD17B10ALDH1A1POLBMAPT
SCHEMBL7743461 0.82 MAPT (0.58) PKMHSD17B10ALDH1A1POLBMAPT
SCHEMBL9372170 0.77 MAPT (0.51) PKMMAPTMEN1KMT2ALMNA
SCHEMBL6956027 0.74 HSD17B10 (0.48) PKMHSD17B10ALDH1A1POLBMAPT
SCHEMBL3286058 0.74 BACE1 (0.36) HSD17B10ALDH1A1MAPTGAACYP1A2
Hydrochloric Acid SCHEMBL9799370 0.72 ALDH1A1 (0.52) PKMHSD17B10ALDH1A1POLBMAPT
SCHEMBL1786217 0.71 HSD17B10 (0.62) PKMHSD17B10ALDH1A1POLBMAPT
SCHEMBL29683253 0.70 GLS (0.61) MEN1KMT2ASMN1; SMN2NPC1RAB9A
SCHEMBL886480 0.70 GLS (0.61) MEN1KMT2ASMN1; SMN2NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0531876-B1 Imidazoindolizine derivatives and process for preparation thereof TANABE SEIYAKU CO (JP) 1996-12-18 EP disclosed
US-5510354-A HYPOTENSIVE AGENTS TANABE SEIYAKU CO., LTD. (JP) 1996-04-23 US disclosed
US-5424316-A Imidazopyridine derivatives for the treatment of hypertension TANABE SEIYAKU CO., LTD. (JP) 1995-06-13 US disclosed
US-5409936-A Useful in prophylaxix; exhibits potent angiotensin ii inhibitory acivities TANABE SEIYAKU CO., LTD. (JP) 1995-04-25 US disclosed
US-5268377-A Imidazoindolizine derivatives process for preparation thereof and use thereof to treat hypertension TANABE SEIYAKU CO., LTD. (JP) 1993-12-07 US disclosed
EP-0531876-A2 Imidazoindolizine derivatives and process for preparation thereof TANABE SEIYAKU CO., LTD. (JP) 1993-03-17 EP disclosed
EP-0531874-A1 Imidazopyridine derivatives and process for preparation thereof TANABE SEIYAKU CO., LTD. (JP) 1993-03-17 EP disclosed