SCHEMBL8992794

SCHEMBL8992794

O=C(O)c1cnc2c(-c3ccc(Cc4ccc5c(c4)OCO5)cc3)cnn2c1O

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.43
KDM4E B2RXH2 3/20 0.43
MAPT P10636 3/20 0.43
NPC1 O15118 2/20 0.43
RAB9A P51151 2/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
NR1H4 Q96RI1 1/20 0.43
KDR P35968 2/20 0.42
RET P07949 3/20 0.41
FYN P06241 2/20 0.41
ABL1 P00519 1/20 0.41
NTRK1 P04629 1/20 0.41
LCK P06239 1/20 0.41
CSF1R P07333 1/20 0.41
PDGFRB P09619 1/20 0.41
PDGFRA P16234 1/20 0.41
FLT1 P17948 1/20 0.41
FLT3 P36888 1/20 0.41
CDK8 P49336 1/20 0.41
NEK2 P51955 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8993204 0.87 SMN1; SMN2 (0.52) ALDH1A1KDM4EMAPTNPC1RAB9A
SCHEMBL8992832 0.83 RAB9A (0.52) ALDH1A1KDM4EMAPTNPC1RAB9A
SCHEMBL8992809 0.81 HSP90AB1 (0.41) ALDH1A1KDM4EMAPTKDRRET
SCHEMBL8993229 0.80 BRS3 (0.52) ALDH1A1KDM4EMAPTNPC1RAB9A
SCHEMBL8992780 0.78 BRS3 (0.54) ALDH1A1KDM4EMAPTNPC1RAB9A
SCHEMBL8993105 0.71 BRS3 (0.45) ALDH1A1KDM4EMAPTNPC1RAB9A
SCHEMBL8993059 0.71 CHEK2 (0.43) ALDH1A1KDRRETLMNACYP1A2
SCHEMBL8992993 0.71 NPC1 (0.68) ALDH1A1KDM4EMAPTNPC1RAB9A
SCHEMBL9165136 0.70 RAB9A (0.52) ALDH1A1KDM4EMAPTNPC1RAB9A
SCHEMBL8992991 0.69 NPC1 (0.57) ALDH1A1KDM4EMAPTNPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5516777-A PROSTATE CANCER THERAPY OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1996-05-14 US disclosed
US-5409928-A Prostate diseases, alopecia OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1995-04-25 US disclosed
EP-0594149-A2 Condensed pyrazole derivatives, method of manufacturing the same, and androgen inhibitor OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1994-04-27 EP disclosed