SCHEMBL8993460

SCHEMBL8993460

CCOC(=S)c1ccc(CC)c(OCCOC)c1Cl

nearest known ligand 0.40

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.32
NPC1 O15118 1/20 0.31
HTT P42858 1/20 0.30
NPSR1 Q6W5P4 1/20 0.30
MEN1 O00255 1/20 0.30
ALDH1A1 P00352 1/20 0.30
CYP1A2 P05177 1/20 0.30
MAPT P10636 1/20 0.30
CYP2C9 P11712 1/20 0.30
CYP2C19 P33261 1/20 0.30
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9194894 0.90 ALDH1A1 (0.31) TSHRALDH1A1
SCHEMBL8993489 0.85 ALDH1A1 (0.34) TSHRNPC1HTTNPSR1MEN1
SCHEMBL9189592 0.84 TSHR (0.32) TSHR
SCHEMBL8993452 0.76 NPC1 (0.33) TSHRNPC1ALDH1A1
SCHEMBL8417857 0.73 CYP4F2 (0.45) TSHRHTTNPSR1MEN1ALDH1A1
SCHEMBL10395568 0.71 ALDH1A1 (0.32) TSHRALDH1A1CYP1A2MAPT
SCHEMBL8993468 0.68 IKBKB (0.42) TSHRHTTMEN1ALDH1A1CYP1A2
SCHEMBL28902378 0.67 METTL3 (0.34) TSHRHTTNPSR1MEN1ALDH1A1
SCHEMBL13490661 0.66 L3MBTL1 (0.46) TSHRNPSR1ALDH1A1MAPTKMT2A
SCHEMBL8993574 0.66 ALDH1A1 (0.44) TSHRALDH1A1MAPTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 13 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0369803-B2 Trisubstituted benzoic acid intermediates ZENECA INC (US) 1996-08-14 EP disclosed
EP-0444152-B1 CERTAIN 2-(2',3',4'-TRISUBSTITUTED BENZOYL)-1,3-CYCLOHEXANEDIONES ZENECA INC (US) 1995-06-14 EP disclosed
EP-0444143-B1 TRISUBSTITUTED BENZOIC ACID INTERMEDIATES ZENECA INC (US) 1994-11-30 EP disclosed
US-5075497-A Chemical intermediate for 2-(2,3,4-trisubstitutedbenzoyl)-1,3-cyclohexanedione ICI AMERICAS, INC. (US) 1991-12-24 US disclosed
US-5073642-A Trisubstituted benzoic acid intermediates ICI AMERICAS INC. (US) 1991-12-17 US disclosed
US-5068423-A Intermediates for herbicides 2-(2,3,4-trisubstituted benzoyl)-1,3-cyclohexanediones ICI AMERICAS INC. (US) 1991-11-26 US disclosed
US-5047572-A For 2-*2,3,4-trisubstituted benzoyl)-1,3-cyclohexanedione ICI AMERICAS INC. (US) 1991-09-10 US disclosed
EP-0444152-A1 CERTAIN 2-(2',3',4'-TRISUBSTITUTED BENZOYL)-1,3-CYCLOHEXANEDIONES. ICI AMERICA INC (US) 1991-09-04 EP disclosed
US-5001256-A Trisubstituted benzoic acid intermediates ICI AMERICAS INC. (US) 1991-03-19 US disclosed
US-4957538-A HERBICIDES ICI AMERICAS INC. (US) 1990-09-18 US disclosed
WO-1990005712-A1 CERTAIN 2-(2',3',4'-TRISUBSTITUTED BENZOYL)-1,3-CYCLOHEXANEDIONES ICI AMERICAS INC. (US) 1990-05-31 WO disclosed
WO-1990005715-A1 TRISUBSTITUTED BENZOIC ACID INTERMEDIATES ICI AMERICAS INC. (US) 1990-05-31 WO disclosed
EP-0369803-A1 Trisubstituted benzoic acid intermediates ZENECA INC. (US) 1990-05-23 EP disclosed