SCHEMBL8993574

SCHEMBL8993574

COCCOc1c(Cl)ccc(C(=O)O)c1Cl

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.44
KDM4E B2RXH2 3/20 0.44
HSD17B10 Q99714 1/20 0.44
PRKAB2 O43741 1/20 0.43
PRKAG1 P54619 1/20 0.43
PRKAA2 P54646 1/20 0.43
PRKAA1 Q13131 1/20 0.43
PRKAG3 Q9UGI9 1/20 0.43
PRKAG2 Q9UGJ0 1/20 0.43
PRKAB1 Q9Y478 1/20 0.43
CLCN2 P51788 2/20 0.40
MAPT P10636 1/20 0.40
TSHR P16473 3/20 0.40
APEX1 P27695 1/20 0.38
HPGD P15428 2/20 0.38
TDP1 Q9NUW8 1/20 0.37
KMT2A Q03164 1/20 0.37
PLAU P00749 1/20 0.36
MAPK1 P28482 1/20 0.36
RARG P13631 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4250810 0.84 TSHR (0.42) ALDH1A1KDM4EHSD17B10CLCN2MAPT
SCHEMBL8417857 0.82 CYP4F2 (0.45) ALDH1A1KDM4EHSD17B10MAPTTSHR
SCHEMBL7976218 0.81 PRKAB2 (0.37) ALDH1A1PRKAB2PRKAG1PRKAA2PRKAA1
SCHEMBL8993484 0.80 PRKAB2 (0.36) ALDH1A1KDM4EPRKAB2PRKAG1PRKAA2
SCHEMBL8993535 0.80 MAPT (0.45) ALDH1A1PRKAB2PRKAG1PRKAA2PRKAA1
SCHEMBL17063591 0.80 ALDH1A1 (0.61) ALDH1A1KDM4EHSD17B10CLCN2MAPT
SCHEMBL9751862 0.78 MAPK1 (0.36) ALDH1A1KDM4EPRKAB2PRKAG1PRKAA2
SCHEMBL3436930 0.77 KMT2A (0.41) ALDH1A1KDM4EHSD17B10KMT2A
SCHEMBL6603561 0.76 KDM4E (0.34) ALDH1A1KDM4EHSD17B10CLCN2TSHR
SCHEMBL24886357 0.76 HPGD (0.45) ALDH1A1KDM4EHSD17B10MAPTAPEX1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0369803-B2 Trisubstituted benzoic acid intermediates ZENECA INC (US) 1996-08-14 EP disclosed
EP-0444152-B1 CERTAIN 2-(2',3',4'-TRISUBSTITUTED BENZOYL)-1,3-CYCLOHEXANEDIONES ZENECA INC (US) 1995-06-14 EP disclosed
EP-0444143-B1 TRISUBSTITUTED BENZOIC ACID INTERMEDIATES ZENECA INC (US) 1994-11-30 EP disclosed
US-5075497-A Chemical intermediate for 2-(2,3,4-trisubstitutedbenzoyl)-1,3-cyclohexanedione ICI AMERICAS, INC. (US) 1991-12-24 US disclosed
US-5073642-A Trisubstituted benzoic acid intermediates ICI AMERICAS INC. (US) 1991-12-17 US disclosed
US-5068423-A Intermediates for herbicides 2-(2,3,4-trisubstituted benzoyl)-1,3-cyclohexanediones ICI AMERICAS INC. (US) 1991-11-26 US disclosed
US-5047572-A For 2-*2,3,4-trisubstituted benzoyl)-1,3-cyclohexanedione ICI AMERICAS INC. (US) 1991-09-10 US disclosed
EP-0444152-A1 CERTAIN 2-(2',3',4'-TRISUBSTITUTED BENZOYL)-1,3-CYCLOHEXANEDIONES. ICI AMERICA INC (US) 1991-09-04 EP disclosed
US-5001256-A Trisubstituted benzoic acid intermediates ICI AMERICAS INC. (US) 1991-03-19 US disclosed
US-4957538-A HERBICIDES ICI AMERICAS INC. (US) 1990-09-18 US disclosed
WO-1990005712-A1 CERTAIN 2-(2',3',4'-TRISUBSTITUTED BENZOYL)-1,3-CYCLOHEXANEDIONES ICI AMERICAS INC. (US) 1990-05-31 WO disclosed
EP-0369803-A1 Trisubstituted benzoic acid intermediates ZENECA INC. (US) 1990-05-23 EP disclosed