SCHEMBL8994002

SCHEMBL8994002

CC(C)Sc1ncc(O)cn1

nearest known ligand 0.36

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 4/20 0.36
ESR2 Q92731 4/20 0.36
HASPIN Q8TF76 2/20 0.34
TSHR P16473 1/20 0.33
PDCD1 Q15116 1/20 0.32
CD274 Q9NZQ7 1/20 0.32
ALDH1A1 P00352 1/20 0.31
LMNA P02545 1/20 0.31
MAPT P10636 1/20 0.31
TDP1 Q9NUW8 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24378472 0.76 MAPT (0.37) HASPINTSHRALDH1A1LMNAMAPT
SCHEMBL5644305 0.76 KDM4E (0.34) HASPINTSHRLMNA
SCHEMBL3281314 0.72 PKM (0.41) HASPINTSHRALDH1A1LMNAMAPT
SCHEMBL850564 0.72
SCHEMBL24378525 0.71 ALDH1A1 (0.39) HASPINALDH1A1
SCHEMBL10814834 0.69
SCHEMBL5609570 0.68 TSHR (0.34) TSHR
SCHEMBL8994058 0.67 APLNR (0.39) ESR1ESR2PDCD1CD274
SCHEMBL12276078 0.65 APLNR (0.43) ESR1ESR2
SCHEMBL17044891 0.65 APLNR (0.43) ESR1ESR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5502190-A DEHYDROHALOGENATION IN THE PRESENCE OF PHASE TRANSFER CATALYST, SOLVENT AND ALKALI METAL HYDROXIDE BAYER CORPORATION (US) 1996-03-26 US disclosed
US-4729987-A Insecticidal O,O-diethyl-O-(2-(1,1-dimethylethyl)-5-pyrimidinyl)-phosphorothioate THE DOW CHEMICAL COMPANY (US) 1988-03-08 US disclosed
US-4654329-A Insecticidal, miticidal or nematocidal phosphorus esters of 5-pyrimidinols THE DOW CHEMICAL COMPANY (US) 1987-03-31 US disclosed
US-4429125-A INSECTICIDES FOR APPLICATION TO SOILS THE DOW CHEMICAL CO. (US) 1984-01-31 US disclosed
EP-0004644-A2 Pyrimidin(5)yl-(thiono)(thiol)-phosphoric(phosphonic) acid esters or amides, process for their preparation and their use as insecticides and acaricides BAYER AG (DE) 1979-10-17 EP disclosed