SCHEMBL8994429

SCHEMBL8994429

O=C(O)C1(Cc2ccccc2)C=NC=CN1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.35
CES2 O00748 1/20 0.33
CES1 P23141 1/20 0.33
AKR1B1 P15121 1/20 0.33
MAPT P10636 2/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
HIF1A Q16665 1/20 0.33
HSD11B1 P28845 1/20 0.32
KEAP1 Q14145 1/20 0.32
MAOA P21397 1/20 0.31
MAOB P27338 1/20 0.31
CYP1A2 P05177 1/20 0.31
ALDH1A1 P00352 1/20 0.31
HCAR2 Q8TDS4 1/20 0.30
TSHR P16473 1/20 0.30
SRR Q9GZT4 1/20 0.30
NPC1 O15118 1/20 0.30
RAB9A P51151 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10998052 0.62
SCHEMBL28079595 0.62 MAOA (0.38) CYP3A4MAPTHSD11B1MAOAMAOB
SCHEMBL28325916 0.60 MAOA (0.32) HSD11B1MAOAMAOBTSHR
SCHEMBL923461 0.60 MAOA (0.48) CES2CES1AKR1B1HSD11B1KEAP1
SCHEMBL28310976 0.59 HSD11B1 (0.36) CYP3A4CES2CES1AKR1B1MAPT
SCHEMBL15122835 0.59 MAOA (0.38) CYP3A4CES2CES1AKR1B1MEN1
SCHEMBL1919144 0.58 SLC6A2 (0.56) MEN1KMT2AHIF1AMAOAMAOB
SCHEMBL3623379 0.58 MAOA (0.41) CES2CES1AKR1B1HSD11B1MAOA
SCHEMBL13818225 0.57 LMNA (0.43) CYP3A4CES2CES1AKR1B1KMT2A
SCHEMBL3716772 0.57 MAOA (0.45) CES2CES1AKR1B1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5512564-A VIRICIDES, AIDS BOEHRINGER MANNHEIM GMBH (DE) 1996-04-30 US disclosed