SCHEMBL8994827

SCHEMBL8994827

Cn1ncnc1-c1ccncc1Cl

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BDKRB2 P30411 2/20 0.43
ATR Q13535 1/20 0.39
PDE2A O00408 1/20 0.38
PDE10A Q9Y233 1/20 0.38
NFATC1 O95644 1/20 0.37
GSK3B P49841 1/20 0.37
DYRK1A Q13627 1/20 0.37
HTT P42858 1/20 0.36
GAA P10253 1/20 0.36
CYP17A1 P05093 4/20 0.35
CYP1A2 P05177 4/20 0.35
ADRA1D P25100 1/20 0.35
ADRA1A P35348 1/20 0.35
ADRA1B P35368 1/20 0.35
KCNH2 Q12809 1/20 0.35
AOC3 Q16853 1/20 0.35
BRD4 O60885 1/20 0.35
LATS1 O95835 1/20 0.33
LATS2 Q9NRM7 1/20 0.33
MAPK8 P45983 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15778938 0.80 ATR (0.44) BDKRB2ATRHTTGAACYP17A1
SCHEMBL8950502 0.80 ADRA1D (0.39) PDE2APDE10ANFATC1GSK3BDYRK1A
SCHEMBL16014644 0.72 CYP3A4 (0.43) BDKRB2HTTGAAADRA1DADRA1A
SCHEMBL31301252 0.71 GSK3B (0.59) NFATC1GSK3BDYRK1AGAAKCNH2
SCHEMBL9007470 0.71 GAA (0.41) DYRK1AHTTGAACYP1A2
SCHEMBL9007469 0.69 CYP2A6 (0.49) HTTGAACYP1A2
SCHEMBL9007472 0.68 CYP1A2 (0.39) HTTGAACYP1A2
SCHEMBL12681315 0.68 SCN9A (0.38) BDKRB2HTTCYP17A1ADRA1DADRA1A
SCHEMBL16583485 0.67 KDM4E (0.37) HTT
SCHEMBL21233156 0.67 CYP11B2 (0.43) BDKRB2HTTGAACYP1A2ADRA1D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8188085-B2 Antifungal agents MERCK SHARP & DOHME CORP. (US) 2012-05-29 US disclosed
US-20100113439-A1 Antifungal agents MERCK & CO., INC. (US) 2010-05-06 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100113439-A1 Antifungal agents GMDS, GBA3, UGGT1 BDKRB2 3739/4885ATR 2294/4885PDE2A 422/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.