SCHEMBL9007472

SCHEMBL9007472

Cn1ncnc1-c1cnccn1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.39
RAB9A P51151 6/20 0.38
P2RX7 Q99572 1/20 0.38
ALDH1A1 P00352 5/20 0.38
TDP1 Q9NUW8 2/20 0.38
GFER P55789 1/20 0.38
RECQL P46063 3/20 0.36
HTT P42858 2/20 0.36
KDM4E B2RXH2 3/20 0.36
CYP3A4 P08684 1/20 0.35
GAA P10253 1/20 0.35
NPC1 O15118 4/20 0.35
MAPT P10636 2/20 0.35
TSHR P16473 2/20 0.35
USP2 O75604 1/20 0.35
PKM P14618 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
HSD17B10 Q99714 1/20 0.35
KMT2A Q03164 2/20 0.35
KDM4A O75164 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8950095 0.77 PIK3CA (0.38) CYP1A2RAB9AP2RX7ALDH1A1TDP1
SCHEMBL15381491 0.73 ALDH1A1 (0.49) CYP1A2RAB9AALDH1A1TDP1RECQL
SCHEMBL30030214 0.73 ALDH1A1 (0.49) CYP1A2RAB9AALDH1A1TDP1RECQL
SCHEMBL21233346 0.72 BRD4 (0.43) CYP1A2RAB9AP2RX7ALDH1A1TDP1
SCHEMBL11126232 0.71 CYP1A2 (0.40) CYP1A2RAB9AP2RX7ALDH1A1TDP1
SCHEMBL3557832 0.70 P2RX7 (0.34) CYP1A2RAB9AP2RX7ALDH1A1TDP1
SCHEMBL9007469 0.70 CYP2A6 (0.49) CYP1A2ALDH1A1HTTKDM4ECYP3A4
SCHEMBL9592630 0.69 CYP11B1 (0.44) CYP1A2RAB9AALDH1A1TDP1GFER
SCHEMBL18912013 0.69 RAB9A (0.51) RAB9AP2RX7ALDH1A1TDP1KDM4E
SCHEMBL11253230 0.68 MAPKAPK2 (0.43) RAB9AALDH1A1TDP1GFERRECQL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8188085-B2 Antifungal agents MERCK SHARP & DOHME CORP. (US) 2012-05-29 US disclosed
US-20100113439-A1 Antifungal agents MERCK & CO., INC. (US) 2010-05-06 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100113439-A1 Antifungal agents GMDS, GBA3, UGGT1 CYP1A2 623/4885RAB9A 1722/4885P2RX7 1931/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.