SCHEMBL8995798

SCHEMBL8995798

CCc1cccc(C)c1C(=O)OC(C)=O

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.41
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
CA7 P43166 1/20 0.41
CA9 Q16790 1/20 0.41
CA14 Q9ULX7 1/20 0.41
GABRA1 P14867 2/20 0.39
GABRB2 P47870 2/20 0.39
NLRP3 Q96P20 2/20 0.39
TAS1R3 Q7RTX0 1/20 0.39
TAS1R1 Q7RTX1 1/20 0.39
TAS1R2 Q8TE23 1/20 0.39
ALDH1A1 P00352 3/20 0.38
TP53 P04637 1/20 0.38
CYP3A4 P08684 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
PTGS2 P35354 1/20 0.37
HSD17B10 Q99714 2/20 0.37
KDM4E B2RXH2 1/20 0.37
HPGD P15428 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5406463 0.85 ALDH1A1 (0.43) CA12CA1CA2CA7CA9
SCHEMBL9881695 0.82 CA12 (0.61) CA12CA1CA2CA7CA9
SCHEMBL10299397 0.82 CA12 (0.52) CA12CA1CA2CA7CA9
SCHEMBL8995835 0.80 CA12 (0.49) CA12CA1CA2CA7CA9
SCHEMBL13105884 0.80 GABRA1 (0.46) CA12CA1CA2CA7CA9
SCHEMBL27340920 0.78 CA12 (0.51) CA12CA1CA2CA7CA9
SCHEMBL28045567 0.77 CD44 (0.41) CA12CA1CA2CA7CA9
SCHEMBL6125235 0.77 MAPT (0.50) ALDH1A1TDP1PTGS2HSD17B10KDM4E
SCHEMBL9833072 0.76 TDP1 (0.45) ALDH1A1TDP1MAOBSMN1; SMN2TSHR
SCHEMBL501450 0.76 GABRA1 (0.46) CA12CA1CA2CA7CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5554617-A Method for treating cancer with 6-aryl pyrimidine compounds THE UPJOHN COMPANY (US) 1996-09-10 US disclosed
US-5434157-A Active against herpes, hepatitis, papovavirus THE UPJOHN COMPANY (US) 1995-07-18 US disclosed
US-5002951-A 2-amino-5-halo-4-pyrimidinol for bactericides and antiprotozoa agent THE UPJOHN COMPANY (US) 1991-03-26 US disclosed
US-4665077-A IMMUNOREGULATORY AGENTS THE UPJOHN COMPANY (US) 1987-05-12 US disclosed
US-4619933-A 6-aryl pyrimidines for treating aplastic anemia THE UPJOHN COMPANY (US) 1986-10-28 US disclosed
US-4543248-A Method for immunoregulation with 6-aryl pyrimidine compounds THE UPJOHN COMPANY (US) 1985-09-24 US disclosed
US-4507302-A Method for treating arthritis with 6-aryl pyrimidine compounds THE UPJOHN COMPANY (US) 1985-03-26 US disclosed