SCHEMBL8995910

SCHEMBL8995910

O=C(C(CCN1CCN(c2cccccc2=O)CC1)c1ccc(Cl)cc1)N1CCCCCC1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 5/20 0.64
HTR1D P28221 1/20 0.64
HTR2B P41595 1/20 0.64
UTS2R Q9UKP6 4/20 0.50
KCNQ2 O43526 1/20 0.44
NTSR1 P30989 1/20 0.43
DRD3 P35462 3/20 0.43
CYP3A4 P08684 2/20 0.43
CYP1A2 P05177 1/20 0.43
CYP2D6 P10635 1/20 0.43
TSHR P16473 1/20 0.43
CYP2C19 P33261 1/20 0.43
HIF1A Q16665 1/20 0.43
SLC22A1 O15245 1/20 0.43
CHRM2 P08172 1/20 0.43
ADRA2A P08913 1/20 0.43
CHRM1 P11229 1/20 0.43
DRD1 P21728 1/20 0.43
TBXA2R P21731 1/20 0.43
SLC6A2 P23975 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8995895 0.92 HTR1A (0.73) HTR1AHTR1DHTR2BKCNQ2CHRM1
SCHEMBL8995908 0.85 HTR1A (0.64) HTR1AHTR1DHTR2BCYP1A2CYP2D6
SCHEMBL8995900 0.81 HTR1A (0.68) HTR1AHTR1DHTR2BKCNQ2DRD3
SCHEMBL8065712 0.78 HTR1A (1.00) HTR1AHTR1DHTR2BCYP3A4CYP1A2
SCHEMBL6546383 0.78 HTR1A (1.00) HTR1AHTR1DHTR2BCYP3A4CYP1A2
SCHEMBL8653841 0.75 HTR1A (0.63) HTR1AHTR1DHTR2BDRD3ADRA1A
SCHEMBL8653834 0.75 HTR1A (0.63) HTR1AHTR1DHTR2BKCNQ2DRD3
SCHEMBL8653021 0.75 HTR1A (0.66) HTR1AHTR1DHTR2BSLC6A4ADRA1A
SCHEMBL8596494 0.75 HTR1A (0.63) HTR1AHTR1DHTR2BADRA1ADRD4
SCHEMBL8652998 0.74 HTR1A (0.62) HTR1AHTR1DHTR2BDRD3KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5541179-A Tropon-2-one piperazine carboxamides as serotonergic agents AMERICAN HOME PRODUCTS CORPORATION (US) 1996-07-30 US disclosed