SCHEMBL8995900

SCHEMBL8995900

COc1cccc(C(CCN2CCN(c3cccccc3=O)CC2)C(=O)N2CCCCCC2)c1

nearest known ligand 0.68

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 3/20 0.68
HTR1D P28221 1/20 0.68
HTR2B P41595 1/20 0.68
DRD4 P21917 7/20 0.52
DRD2 P14416 5/20 0.52
DRD3 P35462 3/20 0.52
OPRM1 P35372 2/20 0.52
KCNQ2 O43526 1/20 0.50
ALDH1A1 P00352 1/20 0.45
LMNA P02545 1/20 0.45
ROCK2 O75116 1/20 0.45
ROCK1 Q13464 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8995895 0.87 HTR1A (0.73) HTR1AHTR1DHTR2BKCNQ2ALDH1A1
SCHEMBL8995908 0.82 HTR1A (0.64) HTR1AHTR1DHTR2BDRD2ALDH1A1
SCHEMBL6546383 0.81 HTR1A (1.00) HTR1AHTR1DHTR2BDRD2ALDH1A1
SCHEMBL8065712 0.81 HTR1A (1.00) HTR1AHTR1DHTR2BDRD2ALDH1A1
SCHEMBL8995910 0.81 HTR1A (0.64) HTR1AHTR1DHTR2BDRD4DRD2
SCHEMBL11106061 0.77 IGF1R (0.55) DRD4DRD2DRD3OPRM1ALDH1A1
SCHEMBL8995919 0.77 NPC1 (0.49) HTR1AHTR1DHTR2BOPRM1KCNQ2
SCHEMBL17206662 0.76 KCNQ2 (0.50) HTR1AHTR1DHTR2BOPRM1KCNQ2
SCHEMBL8654532 0.75 HTR1A (0.64) HTR1AHTR1DHTR2BDRD4DRD2
SCHEMBL8878656 0.74 HTR1A (0.63) HTR1AHTR1DHTR2BDRD4DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5541179-A Tropon-2-one piperazine carboxamides as serotonergic agents AMERICAN HOME PRODUCTS CORPORATION (US) 1996-07-30 US disclosed