SCHEMBL8995908

SCHEMBL8995908

CCOc1ccc(C(CCN2CCN(c3cccccc3=O)CC2)C(=O)N2CCCCCC2)cc1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 3/20 0.64
HTR1D P28221 1/20 0.64
HTR2B P41595 1/20 0.64
DRD2 P14416 1/20 0.46
HTR2A P28223 1/20 0.46
HRH1 P35367 1/20 0.46
KDM4E B2RXH2 2/20 0.45
CYP1A2 P05177 1/20 0.45
GAA P10253 1/20 0.45
CYP2D6 P10635 1/20 0.45
CYP2C9 P11712 1/20 0.45
CYP2C19 P33261 1/20 0.45
MAPK1 P28482 1/20 0.44
MAPT P10636 3/20 0.43
ALDH1A1 P00352 3/20 0.43
LMNA P02545 2/20 0.43
TP53 P04637 2/20 0.43
KMT2A Q03164 2/20 0.43
HPGD P15428 2/20 0.42
HTR7 P34969 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8995895 0.88 HTR1A (0.73) HTR1AHTR1DHTR2BALDH1A1LMNA
SCHEMBL8995910 0.85 HTR1A (0.64) HTR1AHTR1DHTR2BDRD2CYP1A2
SCHEMBL8995900 0.82 HTR1A (0.68) HTR1AHTR1DHTR2BDRD2ALDH1A1
SCHEMBL8065712 0.78 HTR1A (1.00) HTR1AHTR1DHTR2BDRD2HTR2A
SCHEMBL6546383 0.78 HTR1A (1.00) HTR1AHTR1DHTR2BDRD2HTR2A
SCHEMBL8995907 0.75 HPGD (0.56) KDM4EMAPTALDH1A1LMNATP53
SCHEMBL8653021 0.73 HTR1A (0.66) HTR1AHTR1DHTR2BDRD2HTR2A
SCHEMBL8652998 0.72 HTR1A (0.62) HTR1AHTR1DHTR2BDRD2HTR2A
SCHEMBL8653834 0.71 HTR1A (0.63) HTR1AHTR1DHTR2BDRD2HTR2A
SCHEMBL8653841 0.71 HTR1A (0.63) HTR1AHTR1DHTR2BDRD2GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5541179-A Tropon-2-one piperazine carboxamides as serotonergic agents AMERICAN HOME PRODUCTS CORPORATION (US) 1996-07-30 US disclosed