SCHEMBL8996619

SCHEMBL8996619

COC(=O)C[C@H](NC(C)C)C(=O)OC

nearest known ligand 0.38

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.37
CA12 O43570 3/20 0.36
CA1 P00915 2/20 0.36
CA2 P00918 2/20 0.36
CA9 Q16790 2/20 0.36
SMN1; SMN2 Q16637 3/20 0.35
HSD17B10 Q99714 1/20 0.34
MGAM O43451 1/20 0.34
GAA P10253 1/20 0.34
SI P14410 1/20 0.34
MGAM2 Q2M2H8 1/20 0.34
BIRC2 Q13490 1/20 0.34
CA14 Q9ULX7 2/20 0.33
TAS1R3 Q7RTX0 1/20 0.33
TAS1R1 Q7RTX1 1/20 0.33
MAPT P10636 1/20 0.33
RAB9A P51151 1/20 0.33
MME P08473 1/20 0.33
ALDH1A1 P00352 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL752074 1.00 TSHR (0.37) TSHRCA12CA1CA2CA9
SCHEMBL8996690 1.00 TSHR (0.37) TSHRCA12CA1CA2CA9
SCHEMBL20022609 0.89 TSHR (0.42) TSHRCA12CA1CA2CA9
SCHEMBL25475997 0.86 TSHR (0.33) TSHRHSD17B10MGAMGAASI
SCHEMBL2580362 0.84 TSHR (0.44) TSHRCA12CA1CA2CA9
SCHEMBL2580366 0.84 TSHR (0.44) TSHRCA12CA1CA2CA9
SCHEMBL14969737 0.83 ALDH1A1 (0.37) TSHRHSD17B10MGAMGAASI
SCHEMBL19090746 0.82 BIRC2 (0.38) TSHRCA12CA1CA2CA9
SCHEMBL14591443 0.82 CA1 (0.37) TSHRCA12CA1CA2CA9
SCHEMBL20988042 0.80 BIRC2 (0.39) TSHRCA12CA1CA2CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105693634-B Compound and application thereof 清华大学 2018-12-11 CN disclosed
CN-105693634-A Compound and application thereof 清华大学 2016-06-22 CN disclosed
EP-1594843-B1 METHOD FOR PRODUCING AN OPTICALLY ACTIVE beta-amino acid derivative TAKASAGO PERFUMERY CO LTD (JP) 2013-05-22 EP disclosed
US-8188307-B2 Method for producing an optically active tetrahydroquinoline TAKASAGO INTERNATIONAL CORPORATION (JP) 2012-05-29 US disclosed
US-20100036149-A1 METHOD FOR PRODUCING AN OPTICALLY ACTIVE TETRAHYDROQUINOLINE TAKASAGO INTERNATIONAL COPORATION (JP) 2010-02-11 US disclosed
US-7601842-B2 Method for producing an optically active tetrahydroquinoline TAKASAGO INTERNATIONAL CORPORATION (JP) 2009-10-13 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100036149-A1 METHOD FOR PRODUCING AN OPTICALLY ACTIVE TETRAHYDROQUINOLINE AADAT, KMO, ALDH7A1 TSHR 3311/4885CA12 2615/4885CA1 1662/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.