SCHEMBL8996728

SCHEMBL8996728

C[C@H]1[C@@H](Oc2ccc(C#N)cc2)[C@H]2N(C)C(=O)CC[C@]2(C)[C@H]2CC[C@]3(C)CCC[C@H]3[C@H]12

nearest known ligand 0.35

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
TRPC6 Q9Y210 9/20 0.35
HRH3 Q9Y5N1 7/20 0.34
MBOAT4 Q96T53 2/20 0.34
HRH2 P25021 3/20 0.33
HRH1 P35367 3/20 0.33
KCNH2 Q12809 2/20 0.32
SCN5A Q14524 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8523925 1.00 TRPC6 (0.35) TRPC6HRH3MBOAT4HRH2HRH1
SCHEMBL8996718 0.91 SLC6A2 (0.34) MBOAT4HRH1
SCHEMBL8523871 0.91 SLC6A2 (0.34) MBOAT4HRH1
SCHEMBL8996733 0.90 STS (0.30)
SCHEMBL8523662 0.90 STS (0.30)
SCHEMBL8523449 0.89 SRD5A1 (0.33)
SCHEMBL8523677 0.89 STS (0.32)
SCHEMBL8522770 0.89 PLA2G7 (0.33)
SCHEMBL8524175 0.89 SRD5A1 (0.36)
SCHEMBL8523590 0.88 MMP12 (0.33)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0724592-A1 16-SUBSTITUTED-4-AZA-ANDROSTANE 5-ALPHA-REDUCTASE ISOZYME 1 INHIBITORS MERCK & CO. INC. (US) 1996-08-07 EP disclosed
WO-1995011254-A1 16-SUBSTITUTED-4-AZA-ANDROSTANE 5-ALPHA-REDUCTASE ISOZYME 1 INHIBITORS MERCK & CO., INC. (US) 1995-04-27 WO disclosed