SCHEMBL8997199

SCHEMBL8997199

CC#CC(Cc1ccc(C(=O)N[C@@H](CCC(=O)O)C(=O)O)cc1)CC1CNc2nc(N)nc(N)c21

nearest known ligand 0.57

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
DHFR P00374 4/20 0.51
ATIC P31939 3/20 0.49
GART P22102 4/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8997161 0.88 DHFR (0.56) DHFRATICGART
SCHEMBL8997201 0.87 DHFR (0.55) DHFRATICGART
SCHEMBL9397723 0.86 DHFR (0.53) DHFRATICGART
SCHEMBL9039610 0.84 DHFR (0.50) DHFRATICGART
SCHEMBL8997146 0.84 ATIC (0.50) DHFRATICGART
SCHEMBL9041233 0.83 DHFR (0.49) DHFRATICGART
SCHEMBL8997257 0.81 GART (0.61) DHFRATICGART
SCHEMBL9758306 0.79 DHFR (0.55) DHFRATICGART
SCHEMBL8997170 0.79 DHFR (0.55) DHFRATICGART
SCHEMBL9088274 0.79 ATIC (0.51) DHFRATICGART

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0334636-B1 Pyrrolopyrimidine derivatives, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1996-10-23 EP disclosed
US-5539113-A ANTITUMOR AGENTS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-07-23 US disclosed
US-5106974-A Antitumor and -carcinogenic agents TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1992-04-21 US disclosed
US-4997838-A Antitumor agents TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1991-03-05 US disclosed
EP-0334636-A2 Pyrrolopyrimidine derivatives, their production and use Takeda Chemical Industries, Ltd. (JP) 1989-09-27 EP disclosed