SCHEMBL8997146

SCHEMBL8997146

CC#CC(CCC1CNc2nc(N)nc(N)c21)c1ccc(C(=O)N[C@@H](CCC(=O)O)C(=O)O)cc1

nearest known ligand 0.57

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
ATIC P31939 3/20 0.50
GART P22102 5/20 0.47
DHFR P00374 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8997170 0.88 DHFR (0.55) ATICGARTDHFR
SCHEMBL9758306 0.88 DHFR (0.55) ATICGARTDHFR
SCHEMBL8997253 0.86 DHFR (0.58) ATICGARTDHFR
SCHEMBL9397716 0.86 DHFR (0.53) ATICGARTDHFR
SCHEMBL9227822 0.85 DHFR (0.52) ATICGARTDHFR
SCHEMBL9758337 0.84 DHFR (0.60) ATICGARTDHFR
SCHEMBL8997214 0.84 ATIC (0.49) ATICGART
SCHEMBL8997199 0.84 DHFR (0.51) ATICGARTDHFR
SCHEMBL8997198 0.83 ATIC (0.48) ATICGARTDHFR
SCHEMBL9088274 0.82 ATIC (0.51) ATICGARTDHFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5539113-A ANTITUMOR AGENTS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-07-23 US disclosed
US-5106974-A Antitumor and -carcinogenic agents TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1992-04-21 US disclosed
US-4997838-A Antitumor agents TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1991-03-05 US disclosed