SCHEMBL10189208

SCHEMBL10189208

COc1cccc2nc(-c3ccc(-c4ccc(C5CCCCC5)cc4)cn3)[nH]c12

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 3/20 0.42
PDGFRB P09619 1/20 0.37
PDGFRA P16234 1/20 0.37
DGAT1 O75907 4/20 0.35
DHODH Q02127 1/20 0.35
RAF1 P04049 1/20 0.34
MAP4K1 Q92918 3/20 0.34
ALDH1A1 P00352 2/20 0.34
HPGD P15428 2/20 0.34
HSD17B10 Q99714 2/20 0.34
IL2 P60568 2/20 0.34
KDM4E B2RXH2 1/20 0.34
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34
CLK1 P49759 1/20 0.34
HIPK2 Q9H2X6 1/20 0.34
CLK4 Q9HAZ1 1/20 0.34
PDE7A Q13946 1/20 0.34
CDK4 P11802 1/20 0.34
CCND1 P24385 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL900018 0.84 DGAT1 (0.55) DGAT1
SCHEMBL901499 0.77 DGAT1 (0.61) DGAT1
SCHEMBL902206 0.72 DGAT1 (0.61) DGAT1NPC1CBFB
SCHEMBL18790540 0.68 DHODH (0.47) S1PR1DGAT1DHODHRAF1KDM4E
SCHEMBL902783 0.68 DGAT1 (0.45) DGAT1MAP4K1CLK1HIPK2CLK4
SCHEMBL18790847 0.67 NPC1 (0.45) DGAT1DHODHRAF1ALDH1A1KDM4E
SCHEMBL28027631 0.67 TNKS (0.54) ALDH1A1HPGDHSD17B10KDM4ENPC1
SCHEMBL16526751 0.67 S1PR1 (0.53) S1PR1DGAT1DHODHKDM4ENPC1
SCHEMBL5201225 0.66 PDE4A (0.41) ALDH1A1TP53SMN1; SMN2
SCHEMBL25796475 0.63 DHODH (0.40) S1PR1DHODHRAF1S1PR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012044567-A2 IMIDAZOLE DERIVATIVES MERCK SHARP & DOHME CORP. (US) 2012-04-05 WO disclosed