SCHEMBL902393

SCHEMBL902393

COc1cccc2nc(-c3ccc(C4=CC=C(C5CCC(CC(=O)O)CC5)CC4)cc3)[nH]c12

nearest known ligand 0.42

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
DGAT1 O75907 16/20 0.42
SOAT1 P35610 3/20 0.42
KCNH2 Q12809 7/20 0.39
ADORA2A P29274 4/20 0.39
CCNT1 O60563 1/20 0.37
CDK9 P50750 1/20 0.37
HPSE Q9Y251 1/20 0.35
FAAH O00519 1/20 0.35
CHRM2 P08172 1/20 0.35
DGAT2 Q96PD7 1/20 0.35
PDE10A Q9Y233 1/20 0.35
PDE4A P27815 2/20 0.35
PDE4B Q07343 2/20 0.35
PDE4C Q08493 2/20 0.35
PDE4D Q08499 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL901499 0.78 DGAT1 (0.61) DGAT1SOAT1KCNH2ADORA2A
SCHEMBL901617 0.78 DGAT1 (0.50) DGAT1SOAT1KCNH2ADORA2A
SCHEMBL900018 0.77 DGAT1 (0.55) DGAT1SOAT1KCNH2ADORA2A
SCHEMBL10188922 0.73 DGAT1 (0.41) DGAT1SOAT1KCNH2ADORA2A
SCHEMBL6528644 0.71 KDM4E (0.56) ADORA2ACDK9HPSEPDE4APDE4B
SCHEMBL902399 0.71 DGAT1 (0.60) DGAT1SOAT1FAAHCHRM2DGAT2
SCHEMBL10189190 0.70 DGAT1 (0.44) DGAT1SOAT1KCNH2ADORA2A
SCHEMBL902749 0.69 DGAT1 (0.55) DGAT1SOAT1FAAHCHRM2DGAT2
SCHEMBL28027631 0.69 TNKS (0.54) CDK9HPSE
SCHEMBL900619 0.68 DGAT1 (0.56) DGAT1SOAT1FAAHCHRM2DGAT2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012044567-A2 IMIDAZOLE DERIVATIVES MERCK SHARP & DOHME CORP. (US) 2012-04-05 WO disclosed