SCHEMBL9002252

SCHEMBL9002252

O=C(c1cccnc1)c1cccc(C(F)(F)F)c1

nearest known ligand 0.64

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.64
MEN1 O00255 1/20 0.64
KMT2A Q03164 1/20 0.64
VNN1 O95497 10/20 0.64
SRD5A2 P31213 1/20 0.60
CES2 O00748 1/20 0.57
TBXAS1 P24557 2/20 0.56
ALOX15 P16050 1/20 0.56
CASP1 P29466 1/20 0.56
NPSR1 Q6W5P4 1/20 0.56
HSD17B10 Q99714 1/20 0.56
CSF1R P07333 1/20 0.55
BRAF P15056 1/20 0.55
TBXA2R P21731 1/20 0.55
RXFP1 Q9HBX9 1/20 0.53
CNR2 P34972 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10663373 0.89 TSHR (0.55) TSHRMEN1KMT2AVNN1SRD5A2
SCHEMBL10841345 0.88 CES2 (0.72) TSHRMEN1KMT2AVNN1SRD5A2
SCHEMBL1237189 0.85 SRD5A2 (0.79) MEN1KMT2AVNN1SRD5A2CES2
SCHEMBL30706506 0.84 VNN1 (0.60) TSHRMEN1KMT2AVNN1SRD5A2
SCHEMBL15648102 0.84 VNN1 (0.60) TSHRMEN1KMT2AVNN1SRD5A2
SCHEMBL1044812 0.80 SRD5A2 (0.83) VNN1SRD5A2CES2NPSR1CNR2
SCHEMBL18286220 0.79 VNN1 (1.00) VNN1
SCHEMBL1242243 0.79 ALDH1A1 (0.71) MEN1KMT2A
SCHEMBL29915528 0.79 ALDH1A1 (0.71) MEN1KMT2A
SCHEMBL30706504 0.79 AGTR1 (0.57) MEN1KMT2ACES2TBXAS1CSF1R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5482948-A Pyridyl derivatives and pharmaceutical compositions comprising these compounds DR. KARL THOMAE GMBH (DE) 1996-01-09 US disclosed
EP-0547517-B1 Pyridyl derivatives, medicines containing these compounds and processes for their preparation THOMAE GMBH DR K (DE) 1995-05-17 EP disclosed
EP-0547517-A1 Pyridyl derivatives, medicines containing these compounds and processes for their preparation Dr. Karl Thomae GmbH (DE) 1993-06-23 EP disclosed