SCHEMBL9002686

SCHEMBL9002686

O=C(NCCSc1cccc2nccn12)c1ccncc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 5/20 0.43
NPC1 O15118 5/20 0.42
SMN1; SMN2 Q16637 5/20 0.42
NFKB1 P19838 1/20 0.42
NFKB2 Q00653 1/20 0.42
RELA Q04206 1/20 0.42
RECQL P46063 1/20 0.42
MAPT P10636 1/20 0.41
EPHX2 P34913 1/20 0.41
ALDH1A1 P00352 1/20 0.41
KMT2A Q03164 2/20 0.41
MEN1 O00255 1/20 0.41
NAAA Q02083 1/20 0.40
TP53 P04637 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
PKM P14618 1/20 0.39
HTT P42858 1/20 0.39
GFER P55789 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9002351 0.92 RAB9A (0.52) RAB9ANPC1SMN1; SMN2NFKB1NFKB2
SCHEMBL9002081 0.88 RAB9A (0.58) RAB9ANPC1SMN1; SMN2MAPTEPHX2
SCHEMBL9002200 0.84 IDO1 (0.46) RAB9ANPC1SMN1; SMN2NFKB1NFKB2
SCHEMBL9001892 0.83 NPC1 (0.52) RAB9ANPC1SMN1; SMN2MAPTALDH1A1
SCHEMBL9001920 0.83 MTNR1A (0.47) ALDH1A1KMT2A
SCHEMBL9002608 0.83 HPGD (0.41) RAB9ANPC1SMN1; SMN2MAPTALDH1A1
SCHEMBL9002070 0.82 HPGD (0.43) RAB9ANPC1SMN1; SMN2RECQLMAPT
SCHEMBL9001977 0.81 MTNR1B (0.37) RAB9ANPC1SMN1; SMN2NFKB1NFKB2
SCHEMBL9002400 0.81 MTNR1A (0.35) RAB9ANPC1SMN1; SMN2NFKB1NFKB2
Hydrochloric Acid SCHEMBL9001869 0.81 HPGD (0.42) RAB9ANPC1SMN1; SMN2RECQLMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5587383-A CALMODULIN INHIBITORS; ANTIISCHEMIC AGENTS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-12-24 US disclosed
EP-0471236-B1 Imidazopyridine derivatives and their use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1995-03-15 EP disclosed
US-5395839-A Calmodulin and angiogenesis inhibitors TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1995-03-07 US disclosed
US-5244908-A Calmodulin inhibitors TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1993-09-14 US disclosed
EP-0471236-A1 Imidazopyridine derivatives and their use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1992-02-19 EP disclosed