SCHEMBL9001920

SCHEMBL9001920

CC(=O)NCCSc1cccc2nccn12

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 10/20 0.47
MTNR1B P49286 8/20 0.47
TSHR P16473 2/20 0.36
GSTP1 P09211 1/20 0.36
GSTM2 P28161 1/20 0.36
CDK8 P49336 2/20 0.35
ROCK1 Q13464 2/20 0.35
CHEK1 O14757 1/20 0.35
MAP4K4 O95819 1/20 0.35
CSF1R P07333 1/20 0.35
PRKACA P17612 1/20 0.35
KDR P35968 1/20 0.35
MAP2K1 Q02750 1/20 0.35
ACVR1 Q04771 1/20 0.35
MAP4K2 Q12851 1/20 0.35
DYRK1A Q13627 1/20 0.35
AURKB Q96GD4 1/20 0.35
DYRK1B Q9Y463 1/20 0.35
FLT1 P17948 1/20 0.35
CDK9 P50750 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9001977 0.88 MTNR1B (0.37) MTNR1AMTNR1BCDK8ROCK1CHEK1
SCHEMBL9002400 0.88 MTNR1A (0.35) MTNR1AMTNR1BCDK8ROCK1CHEK1
SCHEMBL9002613 0.86 CNR2 (0.37) MTNR1AMTNR1BCDK8ROCK1CHEK1
SCHEMBL9002210 0.86 SMN1; SMN2 (0.38) MTNR1AMTNR1BCDK8ROCK1CHEK1
SCHEMBL9002397 0.84 ALDH1A1 (0.36) MTNR1AMTNR1BTSHRCDK8ROCK1
SCHEMBL9002309 0.84 SMN1; SMN2 (0.37) CDK8ROCK1FLT1CDK9LIMK1
SCHEMBL9002005 0.84 HTT (0.43) TSHRCDK8ALDH1A1
SCHEMBL9002351 0.84 RAB9A (0.52) ALDH1A1KMT2AL3MBTL1
SCHEMBL9002790 0.84 ALDH1A1 (0.33) MTNR1AMTNR1BCDK8ROCK1CHEK1
Hydrochloric Acid SCHEMBL9001885 0.84 NPC1 (0.39) MTNR1AMTNR1BCDK8ROCK1CHEK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5587383-A CALMODULIN INHIBITORS; ANTIISCHEMIC AGENTS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-12-24 US disclosed
EP-0471236-B1 Imidazopyridine derivatives and their use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1995-03-15 EP disclosed
US-5395839-A Calmodulin and angiogenesis inhibitors TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1995-03-07 US disclosed
US-5244908-A Calmodulin inhibitors TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1993-09-14 US disclosed
EP-0471236-A1 Imidazopyridine derivatives and their use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1992-02-19 EP disclosed