SCHEMBL9004046

SCHEMBL9004046

COc1c(C)cc(C(C)=O)cc1C(=O)O

nearest known ligand 0.46

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 3/20 0.46
LMNA P02545 1/20 0.43
AKR1C3 P42330 10/20 0.43
AKR1C2 P52895 10/20 0.43
KDM4E B2RXH2 3/20 0.41
ALDH1A1 P00352 3/20 0.41
HPGD P15428 3/20 0.41
TPMT P51580 2/20 0.39
MAPT P10636 1/20 0.39
TDP1 Q9NUW8 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27801015 0.89 TPMT (0.49) HSD17B10KDM4EALDH1A1HPGDTPMT
SCHEMBL2796551 0.85 LMNA (0.52) LMNAALDH1A1TPMTMAPT
SCHEMBL11111361 0.82 LMNA (0.56) HSD17B10LMNAAKR1C3AKR1C2KDM4E
SCHEMBL1434189 0.81 HSD17B10 (0.52) HSD17B10KDM4EALDH1A1HPGDTPMT
SCHEMBL11618007 0.80 ATM (0.47) HSD17B10LMNAAKR1C3KDM4EALDH1A1
SCHEMBL10920134 0.79 KDM4E (0.55) HSD17B10AKR1C3AKR1C2KDM4EALDH1A1
SCHEMBL11617870 0.79 THRA (0.44) HSD17B10KDM4EALDH1A1HPGDTDP1
SCHEMBL19100974 0.78 HSD17B10 (0.49) HSD17B10KDM4EALDH1A1HPGDMAPT
SCHEMBL786462 0.78 LMNA (0.60) LMNAKDM4EALDH1A1HPGDTPMT
SCHEMBL2978683 0.78 LMNA (0.50) HSD17B10LMNAKDM4EALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0733037-A1 ARYL SUBSTITUTED AMINO ACIDS, CNS INFLUENCING AGENTS UNIVERSITY OF BRISTOL (GB) 1996-09-25 EP disclosed
WO-1995015941-A1 ARYL SUBSTITUTED AMINO ACIDS, CNS INFLUENCING AGENTS UNIVERSITY OF BRISTOL (GB) 1995-06-15 WO disclosed
US-4301159-A FOR GASTRIC DISORDERS, ANTIEMETICS SHIONOGI & CO., LTD. (JP) 1981-11-17 US disclosed
US-4127666-A ANTIEMETIC UNIVERSITE D'ORLEANS (FR) 1978-11-28 US disclosed